SCHEMBL2833598

SCHEMBL2833598

CCn1nc(-c2nc(-c3ccc(C(N)=O)cc3C3CC3)no2)c2c1CC(C)(C)CC2.CCn1nc(-c2nc(-c3ccc(N)nc3C(F)(F)F)no2)c2c1CC(C)(C)CC2

nearest known ligand 0.31

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 3/20 0.31
HSP90AB1 P08238 2/20 0.31
HSP90B1 P14625 1/20 0.31
TRAP1 Q12931 1/20 0.31
HDAC4 P56524 1/20 0.30
S1PR1 P21453 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3463052 0.91 CYP2D6 (0.33) HSP90AA1HSP90AB1S1PR1
SCHEMBL2474054 0.88 ALOX5AP (0.31)
SCHEMBL2473825 0.85 RARB (0.38) HDAC4S1PR1
SCHEMBL3462797 0.85 S1PR1 (0.38) S1PR1
SCHEMBL2472183 0.83 OPRM1 (0.36) S1PR1
SCHEMBL3462877 0.82 S1PR1 (0.36) HSP90AA1HSP90AB1S1PR1
SCHEMBL2527579 0.80 HDAC4 (0.30) HDAC4
SCHEMBL2474605 0.78 RARB (0.45) HDAC4S1PR1
SCHEMBL2474311 0.77 NPC1 (0.39) HSP90AA1HSP90AB1HDAC4S1PR1
SCHEMBL2476261 0.76 RARB (0.37) HDAC4S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010072352-A1 1, 2, 4 -OXADIAZOLE DERIVATIVES AND THEIR THERAPEUTIC USE ALMIRALL S.A. (ES) 2010-07-01 WO claimed