SCHEMBL28337477

SCHEMBL28337477

Clc1ccc2c(ccn2-c2ncccn2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KA5 O75582 6/20 0.47
RPS6KA4 O75676 2/20 0.45
ROCK1 Q13464 3/20 0.43
CDC7 O00311 1/20 0.43
CDK2 P24941 1/20 0.43
MAP3K14 Q99558 1/20 0.43
BIRC5 O15392 1/20 0.42
ROCK2 O75116 1/20 0.41
PIM1 P11309 1/20 0.41
PIM3 Q86V86 1/20 0.41
NR4A2 P43354 1/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
SLC6A2 P23975 1/20 0.39
CYP19A1 P11511 1/20 0.38
FGFR1 P11362 1/20 0.38
HPGD P15428 1/20 0.36
OXER1 Q8TDS5 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HCRTR1 O43613 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29388268 0.82 ROCK1 (0.47) RPS6KA5ROCK1CDC7CDK2MAP3K14
SCHEMBL28307170 0.82 ROCK1 (0.47) RPS6KA5ROCK1CDC7CDK2MAP3K14
SCHEMBL29961473 0.79 MAPT (0.49) RPS6KA5RPS6KA4ROCK1CDC7CDK2
SCHEMBL31735756 0.79 PRKCI (0.49) RPS6KA5RPS6KA4ROCK1CDC7CDK2
SCHEMBL28901206 0.79 RPS6KA5 (0.51) RPS6KA5RPS6KA4ROCK1CDC7CDK2
SCHEMBL28371918 0.79 ROCK1 (0.57) RPS6KA5RPS6KA4ROCK1HTR2AHTR2C
SCHEMBL7914102 0.79 ROCK1 (0.57) RPS6KA5RPS6KA4ROCK1CDC7CDK2
SCHEMBL28370777 0.79 MAPT (0.49) RPS6KA5RPS6KA4ROCK1CDC7CDK2
SCHEMBL20647687 0.79 ROCK2 (0.36) RPS6KA5ROCK1CDC7CDK2MAP3K14
SCHEMBL17671266 0.76 MEN1 (0.38) CDC7ROCK2PIM1PIM3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109678810-B 1,2-oxygen nitrogen heterocyclic butane compound and preparation method and application thereof 南京工业大学 2022-10-28 CN claimed
CN-109678810-B 1,2-oxygen nitrogen heterocyclic butane compound and preparation method and application thereof 南京工业大学 2022-10-28 CN disclosed
CN-106279236-B Method for synthesizing 2-triisopropyl silicon-based acetylene indole compound 南京理工大学 2020-04-10 CN disclosed
CN-110563701-A N-2-pyrimidine-2-azido-3- (2,2,6, 6-tetramethylpiperidinyloxy) indoline and preparation and application thereof 浙江工业大学 2019-12-13 CN disclosed