SCHEMBL28344280

SCHEMBL28344280

CCOC(=O)c1cc(Cl)c(CBr)n(-c2ccc(F)cc2)c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MAPK1 P28482 1/20 0.46
CYP4F2 P78329 1/20 0.46
CYP4A11 Q02928 1/20 0.46
CHRNA7 P36544 2/20 0.44
ALDH1A1 P00352 4/20 0.44
HSD17B10 Q99714 2/20 0.44
TP53 P04637 1/20 0.44
HPGD P15428 1/20 0.44
POLB P06746 1/20 0.42
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
BAZ2B Q9UIF8 1/20 0.41
BAZ2A Q9UIF9 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PKM P14618 1/20 0.41
CYP1A2 P05177 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28880873 0.90 KDM4E (0.48) KDM4ESMN1; SMN2MAPK1CHRNA7ALDH1A1
SCHEMBL28344297 0.89 KDM4E (0.47) KDM4ESMN1; SMN2MAPK1CHRNA7ALDH1A1
SCHEMBL21776585 0.87 CHRNA7 (0.47) KDM4ESMN1; SMN2MAPK1CHRNA7ALDH1A1
SCHEMBL23617168 0.86 KDM4E (0.47) KDM4ESMN1; SMN2MAPK1CHRNA7ALDH1A1
SCHEMBL28341774 0.86 MAPK1 (0.53) KDM4ESMN1; SMN2MAPK1CHRNA7ALDH1A1
SCHEMBL28344369 0.84 KDM4E (0.51) KDM4ESMN1; SMN2MAPK1CHRNA7ALDH1A1
SCHEMBL28344699 0.83 KDM4E (0.48) KDM4ESMN1; SMN2MAPK1CHRNA7ALDH1A1
SCHEMBL28344292 0.82 KDM4E (0.47) KDM4ESMN1; SMN2MAPK1CHRNA7ALDH1A1
SCHEMBL28342007 0.82 KDM4E (0.50) KDM4ESMN1; SMN2MAPK1CHRNA7ALDH1A1
SCHEMBL28344303 0.81 KDM4E (0.41) KDM4ESMN1; SMN2MAPK1CHRNA7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110627796-B Nitrogenous heterocyclic derivative and application thereof in medicine 北京越之康泰生物医药科技有限公司 2022-07-12 CN disclosed
CN-110627796-A Nitrogenous heterocyclic derivative and application thereof in medicine 北京越之康泰生物医药科技有限公司 2019-12-31 CN disclosed