SCHEMBL28346851

SCHEMBL28346851

CC#CCN1c2c(n(C)c(=O)[nH]c2=O)N(C(C)c2cccc(NC(C)=O)c2)C1N1CCC[C@@H](N)C1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.39
SLC9A3 P48764 1/20 0.39
DPP4 P27487 19/20 0.36
GPR119 Q8TDV5 1/20 0.35
CHRM1 P11229 2/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15533388 0.72 DPP4 (0.47) DPP4
SCHEMBL15533861 0.70 DPP4 (0.43) DPP4KCNH2
SCHEMBL15533174 0.69 DPP4 (0.53) DPP4CHRM1KCNH2
SCHEMBL160189 0.69 DPP4 (0.53) DPP4CHRM1KCNH2
SCHEMBL7533607 0.69 DPP4 (0.36) DPP4CHRM1KCNH2
SCHEMBL15091721 0.67 DPP4 (0.34) DPP4
SCHEMBL27944319 0.66 DPP4 (0.40) DPP4CHRM1
SCHEMBL27600222 0.62 TSHR (0.39) DPP4KCNH2
SCHEMBL6674520 0.61 DPP4 (0.42) CYP2D6DPP4KCNH2
SCHEMBL555775 0.57 ATM (0.35) DPP4CHRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108299436-B Xanthine compound and pharmaceutical composition and application thereof 上海慈瑞医药科技股份有限公司 2020-01-17 CN claimed
CN-108299436-B Xanthine compound and pharmaceutical composition and application thereof 上海慈瑞医药科技股份有限公司 2020-01-17 CN disclosed