SCHEMBL28347246

SCHEMBL28347246

CC(C)Sc1sc(-n2nc(O)c(Br)c2C(=O)O)nc1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 2/20 0.36
MYC P01106 1/20 0.34
WDR5 P61964 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33
DHODH Q02127 1/20 0.33
GRIA4 P48058 1/20 0.33
KDM4E B2RXH2 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ALOX5 P09917 2/20 0.33
PTGS2 P35354 2/20 0.33
ALDH1A1 P00352 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MAPT P10636 2/20 0.32
HSP90AA1 P07900 1/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
BCHE P06276 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20214050 0.90 KDM4E (0.35) PTGER1MYCWDR5PTGDR2DHODH
SCHEMBL29580277 0.84 PTGER1 (0.38) PTGER1KDM4EMEN1KMT2APTGS2
SCHEMBL20224694 0.84 PTGER1 (0.37) PTGER1KDM4EMEN1KMT2AALDH1A1
SCHEMBL20214266 0.84 PTGER1 (0.38) PTGER1KDM4EMEN1KMT2APTGS2
SCHEMBL18295289 0.82 GRIA4 (0.36) PTGER1MYCWDR5DHODHGRIA4
SCHEMBL18282149 0.82 ALDH1A1 (0.34) PTGER1MYCWDR5DHODHKDM4E
SCHEMBL29231587 0.81 PTGER1 (0.38) PTGER1MYCWDR5PTGDR2DHODH
SCHEMBL18282156 0.81 NPC1 (0.37) PTGER1MYCWDR5PTGDR2DHODH
SCHEMBL20214527 0.80 F2RL3 (0.33) PTGER1MYCWDR5DHODHKDM4E
SCHEMBL18282046 0.80 PTGER1 (0.35) PTGER1MYCWDR5PTGDR2DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110603254-B Substituted pyrazole compounds and methods of using the same for treating hyperproliferative diseases 班塔姆制药有限责任公司 2024-04-12 CN disclosed
CN-110603254-A Substituted pyrazole compounds and methods of using the same for treating hyperproliferative diseases 班塔姆制药有限责任公司 2019-12-20 CN disclosed