SCHEMBL28348956

SCHEMBL28348956

C=C1CCC[C@@H](OC(=O)NC(C)(C)C)C1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.36
EPHX1 P07099 2/20 0.35
CCNE1 P24864 4/20 0.32
CDK2 P24941 4/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
GSK3B P49841 3/20 0.32
NTMT1 Q9BV86 1/20 0.32
LMNA P02545 1/20 0.30
NPC1 O15118 1/20 0.30
HTT P42858 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28348910 0.83 THRB (0.42) DPP4EPHX1CCNE1CDK2SMN1; SMN2
SCHEMBL28457660 0.79 EPHX1 (0.38) DPP4EPHX1SMN1; SMN2NPC1HTT
SCHEMBL12669754 0.78 EPHX1 (0.48) DPP4EPHX1SMN1; SMN2NTMT1LMNA
SCHEMBL7812041 0.78 EPHX1 (0.53) DPP4EPHX1SMN1; SMN2NPC1HTT
SCHEMBL22105022 0.78 HPGD (0.32) EPHX1
SCHEMBL25270841 0.77 EPHX1 (0.39) DPP4EPHX1CCNE1CDK2SMN1; SMN2
SCHEMBL8495444 0.77 EPHX1 (0.56) DPP4EPHX1SMN1; SMN2NPC1HTT
SCHEMBL7815595 0.74 EPHX1 (0.42) DPP4EPHX1CCNE1CDK2SMN1; SMN2
SCHEMBL22105320 0.73 CYP19A1 (0.31)
SCHEMBL25277512 0.72 EPHX1 (0.36) DPP4EPHX1CCNE1CDK2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105849099-B Polycyclic inhibitors of cyclin dependent kinase 7(CDK7) 达纳-法伯癌症研究所股份有限公司 2020-01-17 CN disclosed