SCHEMBL28349237

SCHEMBL28349237

CSc1ccccc1NC(=O)c1ccc(Br)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.68
KMT2A Q03164 2/20 0.68
NPSR1 Q6W5P4 1/20 0.68
HSD17B10 Q99714 1/20 0.68
ALDH1A1 P00352 4/20 0.65
MAPT P10636 2/20 0.65
L3MBTL1 Q9Y468 4/20 0.58
RAB9A P51151 3/20 0.58
POLB P06746 1/20 0.58
ALOX15 P16050 1/20 0.58
HTT P42858 1/20 0.58
HDAC1 Q13547 1/20 0.57
HDAC8 Q9BY41 1/20 0.57
HDAC6 Q9UBN7 1/20 0.57
NPC1 O15118 1/20 0.55
TDP1 Q9NUW8 2/20 0.55
LMNA P02545 1/20 0.54
MAPK1 P28482 1/20 0.54
TSHR P16473 1/20 0.52
MDM4 O15151 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28399871 0.85 KMT2A (0.69) TP53KMT2ANPSR1HSD17B10ALDH1A1
SCHEMBL97400 0.84 KMT2A (0.68) TP53KMT2ANPSR1HSD17B10ALDH1A1
SCHEMBL23657637 0.84 HDAC1 (0.72) TP53KMT2ANPSR1HSD17B10ALDH1A1
SCHEMBL28346556 0.84 KMT2A (0.72) TP53KMT2ANPSR1HSD17B10ALDH1A1
SCHEMBL28348690 0.84 KMT2A (0.68) TP53KMT2ANPSR1HSD17B10ALDH1A1
SCHEMBL28403540 0.81 F10 (0.77) TP53KMT2ANPSR1HSD17B10ALDH1A1
SCHEMBL11440529 0.80 HPGD (0.74) KMT2ANPSR1HSD17B10ALDH1A1L3MBTL1
SCHEMBL28348662 0.79 ALDH1A1 (1.00) TP53KMT2ANPSR1HSD17B10ALDH1A1
SCHEMBL30608697 0.78 NPC1 (0.70) TP53KMT2ARAB9APOLBHTT
SCHEMBL651227 0.78 NPC1 (0.70) TP53KMT2ARAB9APOLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109369504-B Preparation method of sulfur-containing 3-methylene isoindoline-1-ketone derivative 温州大学 2020-05-12 CN disclosed
CN-107488139-B Preparation method of sulfur-containing 3-arylmethylene isoindolinone derivative WENZHOU UNIVERSITY (CN) 2019-12-10 CN disclosed