SCHEMBL28349986

SCHEMBL28349986

Cn1c(=O)n(CCc2ccccc2)c(=O)c2c1nc(N1CCC[C@@H](N)C1)n2CC#CCF

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.71
CHRM1 P11229 4/20 0.65
POU2F2 P09086 1/20 0.61
ADORA3 P0DMS8 1/20 0.61
POU2F1 P14859 1/20 0.61
CHRM3 P20309 1/20 0.61
HRH2 P25021 1/20 0.61
MC4R P32245 1/20 0.61
FAP Q12884 1/20 0.61
DPP8 Q6V1X1 1/20 0.61
DPP9 Q86TI2 1/20 0.61
GHSR Q92847 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL556151 0.92 DPP4 (0.77) DPP4CHRM1POU2F2ADORA3POU2F1
SCHEMBL28346678 0.92 DPP4 (0.77) DPP4CHRM1POU2F2ADORA3POU2F1
SCHEMBL28752138 0.90 DPP4 (0.82) DPP4CHRM1POU2F2ADORA3POU2F1
SCHEMBL556428 0.89 DPP4 (0.82) DPP4CHRM1POU2F2ADORA3POU2F1
SCHEMBL555576 0.86 DPP4 (0.76) DPP4CHRM1POU2F2ADORA3POU2F1
SCHEMBL28347270 0.86 DPP4 (0.68) DPP4CHRM1POU2F2ADORA3POU2F1
SCHEMBL555521 0.85 DPP4 (0.85) DPP4CHRM1CHRM3
SCHEMBL3968118 0.84 DPP4 (0.83) DPP4CHRM1POU2F2ADORA3POU2F1
SCHEMBL3968112 0.84 DPP4 (0.83) DPP4CHRM1POU2F2ADORA3POU2F1
SCHEMBL555925 0.84 DPP4 (0.81) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108299436-B Xanthine compound and pharmaceutical composition and application thereof 上海慈瑞医药科技股份有限公司 2020-01-17 CN disclosed