SCHEMBL28354491

SCHEMBL28354491

CC(C)(C)OC(=O)NCCOc1ccc(OC(F)(F)F)c(F)c1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.54
CA12 O43570 5/20 0.53
CA1 P00915 5/20 0.53
CA2 P00918 5/20 0.53
CA9 Q16790 5/20 0.53
SCN9A Q15858 1/20 0.44
EPHX2 P34913 1/20 0.43
AAK1 Q2M2I8 2/20 0.41
ITK Q08881 2/20 0.41
EGFR P00533 1/20 0.41
BCHE P06276 1/20 0.41
CNR2 P34972 1/20 0.41
IDO1 P14902 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21601198 0.85 CA12 (0.60) PDK2CA12CA1CA2CA9
SCHEMBL1683350 0.84 CA12 (0.64) PDK2CA12CA1CA2CA9
SCHEMBL28350739 0.83 PDK2 (0.56) PDK2CA12CA1CA2CA9
SCHEMBL29509110 0.82 CA12 (0.56) PDK2CA12CA1CA2CA9
SCHEMBL18290008 0.82 CA12 (0.56) PDK2CA12CA1CA2CA9
SCHEMBL21601185 0.81 CA12 (0.57) PDK2CA12CA1CA2CA9
SCHEMBL28351078 0.81 PPARA (0.53) PDK2CA12CA1CA2CA9
SCHEMBL7428314 0.79 SCN9A (0.53) PDK2CA12CA1CA2CA9
SCHEMBL22809649 0.79 PDK2 (0.45) PDK2SCN9AEPHX2
SCHEMBL3585001 0.79 CA12 (0.67) PDK2CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110612285-B Amide derivatives as Nav1.7 and Nav1.8 blockers 拉夸里亚创药株式会社 2023-04-04 CN disclosed
CN-110612285-A Amide derivatives as Nav1.7 and Nav1.8 blockers 拉夸里亚创药株式会社 2019-12-24 CN disclosed