SCHEMBL22809649

SCHEMBL22809649

CNCCOc1ccc(OC(F)(F)F)c(F)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 2/20 0.45
HTR1B P28222 2/20 0.44
HTR1D P28221 1/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
EPHX2 P34913 1/20 0.42
SLC7A5 Q01650 1/20 0.41
PDE2A O00408 1/20 0.40
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
SCN9A Q15858 1/20 0.38
FFAR4 Q5NUL3 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22809574 0.81 SLC7A5 (0.50) PDK2KDM4EEPHX2SLC7A5PDE2A
Hydrochloric Acid SCHEMBL28350715 0.80 SLC7A5 (0.49) PDK2KDM4EEPHX2SLC7A5PDE2A
Hydrochloric Acid SCHEMBL30450035 0.80 SLC7A5 (0.49) PDK2KDM4EEPHX2SLC7A5PDE2A
SCHEMBL23067893 0.79 HTR1B (0.53) PDK2HTR1BHTR1DKDM4EALDH1A1
SCHEMBL30756577 0.79 HTR1B (0.53) PDK2HTR1BHTR1DKDM4EALDH1A1
SCHEMBL5535001 0.79 HTR1B (0.58) PDK2HTR1BHTR1DKDM4EALDH1A1
SCHEMBL28354491 0.79 PDK2 (0.54) PDK2EPHX2SCN9A
SCHEMBL18295382 0.78 HTR1B (0.52) PDK2HTR1BHTR1DKDM4EALDH1A1
SCHEMBL22809553 0.77 HTR1B (0.56) PDK2HTR1BHTR1DKDM4EALDH1A1
SCHEMBL22208515 0.77 SLC7A5 (0.43) EPHX2SLC7A5PDE2ASCN9AFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3487839-B1 AMIDE DERIVATIVES AS NAV1.7 AND NAV1.8 BLOCKERS RAQUALIA PHARMA INC (JP) 2020-12-23 EP disclosed