SCHEMBL28355432

SCHEMBL28355432

O=C(O)c1ccc(C(=O)NC23CC4CC(CC(C4)C2)C3)cc1

nearest known ligand 0.78

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FAAH O00519 4/20 0.78
CNR2 P34972 5/20 0.76
POLB P06746 1/20 0.73
EPHX2 P34913 3/20 0.68
EPHX1 P07099 2/20 0.59
PKM P14618 1/20 0.58
TSHR P16473 2/20 0.58
ALDH1A1 P00352 2/20 0.58
KDM4E B2RXH2 1/20 0.58
MAPT P10636 1/20 0.58
HPGD P15428 1/20 0.58
ALOX12 P18054 1/20 0.58
HTT P42858 1/20 0.58
ATM Q13315 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
HSD17B10 Q99714 1/20 0.58
LMNA P02545 1/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1421026 0.88 FAAH (1.00) FAAHCNR2POLBEPHX2EPHX1
SCHEMBL2917775 0.86 CNR2 (1.00) FAAHCNR2POLBEPHX2EPHX1
SCHEMBL22308141 0.85 FAAH (0.82) FAAHCNR2POLBEPHX2EPHX1
SCHEMBL7122051 0.85 POLB (1.00) FAAHCNR2POLBEPHX1PKM
SCHEMBL11450782 0.85 CNR2 (0.73) FAAHCNR2POLBPKMTSHR
SCHEMBL19736415 0.82 CNR2 (0.76) FAAHCNR2POLBEPHX2EPHX1
SCHEMBL21292793 0.82 CNR2 (0.69) FAAHCNR2POLBEPHX1PKM
SCHEMBL21309851 0.82 CNR2 (0.69) FAAHCNR2POLBEPHX1PKM
SCHEMBL2913054 0.82 FAAH (0.71) FAAHCNR2POLBEPHX2EPHX1
SCHEMBL16872821 0.81 FAAH (0.71) FAAHCNR2POLBEPHX2EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110759889-B 2-aryl amido substituted thiophene imide ester compound and preparation method and application thereof 中国医学科学院药物研究所 2022-05-20 CN disclosed
CN-110759889-A 2-aryl amido substituted thiophene imide ester compound and preparation method and application thereof 中国医学科学院药物研究所 2020-02-07 CN disclosed