SCHEMBL28355490

SCHEMBL28355490

COc1ccc(C(C2CCNCC2)N2CCC(O)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.46
CHRM1 P11229 1/20 0.46
CACNA2D1 P54289 1/20 0.44
CACNA1B Q00975 1/20 0.44
CACNB1 Q02641 1/20 0.44
OPRM1 P35372 2/20 0.41
OPRD1 P41143 2/20 0.41
OPRK1 P41145 1/20 0.41
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
ADRB1 P08588 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HSD11B1 P28845 2/20 0.39
MMP1 P03956 1/20 0.39
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29785696 0.89 POLB (0.43) CHRM2CHRM1CACNA2D1CACNA1BCACNB1
SCHEMBL28788132 0.89 POLB (0.43) CHRM2CHRM1CACNA2D1CACNA1BCACNB1
SCHEMBL29785758 0.84 ACHE (0.40) CACNA2D1CACNA1BCACNB1OPRM1OPRD1
SCHEMBL28355931 0.84 ACHE (0.40) CACNA2D1CACNA1BCACNB1OPRM1OPRD1
SCHEMBL28944933 0.78 SLC6A4 (0.49) CACNA2D1CACNA1BCACNB1OPRM1OPRD1
SCHEMBL29785705 0.76 SLC6A2 (0.55) CACNA2D1CACNA1BCACNB1SLC6A2SLC6A4
SCHEMBL28788134 0.76 SLC6A2 (0.55) CACNA2D1CACNA1BCACNB1SLC6A2SLC6A4
SCHEMBL5488053 0.76 CXCR4 (0.46) CHRM2CHRM1CACNA2D1CACNA1BCACNB1
SCHEMBL28788127 0.74 SMAD3 (0.42) CHRM2CACNA2D1CACNA1BCACNB1OPRM1
SCHEMBL21788564 0.74 TDP1 (0.47) HTR3EHTR3BADRB1HTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110467597-B Aralkyl cyclamine derivatives and application thereof in multi-target anti-depression drugs 上海医药工业研究院 2022-07-12 CN disclosed
CN-110467597-A Aralkyl cyclammonium analog derivative and its application in multiple target point anti-depression drug SHANGHAI INST PHARMACEUTICAL IND 2019-11-19 CN disclosed