SCHEMBL28358019

SCHEMBL28358019

Cc1cn[c]c(-c2ncccc2C)c1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.45
METAP2 P50579 1/20 0.41
CCR1 P32246 1/20 0.37
CCR5 P51681 1/20 0.37
CCR8 P51685 1/20 0.37
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
CNR2 P34972 1/20 0.35
PLAU P00749 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HRH3 Q9Y5N1 1/20 0.32
SMO Q99835 5/20 0.32
CRHR1 P34998 1/20 0.32
ABL1 P00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28358297 0.77 CCR1 (0.34) CCR1CCR5CCR8
SCHEMBL28361808 0.75 KDM4E (0.43) CYP2A6METAP2CCR1CCR5CCR8
SCHEMBL196235 0.71 CYP2A6 (0.61) CYP2A6METAP2NOS3NOS1NOS2
SCHEMBL29924154 0.71 CYP2A6 (0.61) CYP2A6METAP2NOS3NOS1NOS2
SCHEMBL31252534 0.71 CYP2A6 (0.61) CYP2A6METAP2NOS3NOS1NOS2
SCHEMBL938744 0.70 ALDH1A1 (0.40) CYP2A6METAP2CCR1CCR8NOS3
SCHEMBL12002555 0.69 CYP2A6 (0.43) CYP2A6METAP2NOS3NOS1NOS2
SCHEMBL6118799 0.69 CCR1 (0.55) CYP2A6METAP2CCR1CCR5CCR8
SCHEMBL12320090 0.67 CYP2A6 (0.48) CYP2A6METAP2CCR1CCR8NOS3
SCHEMBL28235663 0.67 CYP2A6 (0.58) CYP2A6METAP2NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110669052-A Substituted 2-azabicyclic compounds and their use as orexin receptor modulators 詹森药业有限公司 2020-01-10 CN disclosed