SCHEMBL28358264

SCHEMBL28358264

Cc1cnc(-c2[c]nccc2)c(F)c1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.36
CCR5 P51681 2/20 0.36
CCR8 P51685 2/20 0.36
KMT2A Q03164 1/20 0.35
PDK2 Q15119 1/20 0.33
CYP1A2 P05177 1/20 0.33
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
DHODH Q02127 1/20 0.30
HTR1A P08908 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2589450 0.78 GABRG2 (0.37) KMT2A
SCHEMBL28358021 0.72 CYP1A2 (0.32) CYP1A2
SCHEMBL28358188 0.72 CYP2A6 (0.31) CCR1CCR5CCR8
SCHEMBL28852322 0.71 CCR1 (0.52) CCR1CCR5CCR8
SCHEMBL28852324 0.68 CCR1 (0.55) CCR1CCR5CCR8KMT2A
SCHEMBL4909130 0.67
SCHEMBL28358102 0.67 KMT2A (0.30) KMT2A
SCHEMBL14635181 0.67 NAMPT (0.33)
SCHEMBL24602339 0.66 RPS6KA3 (0.45) CCR1CCR5CCR8KMT2APTGS2
SCHEMBL1515426 0.66 NISCH (0.38) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110669052-B Substituted 2-azabicyclic compounds and their use as orexin receptor modulators 詹森药业有限公司 2022-10-11 CN disclosed
CN-110669052-A Substituted 2-azabicyclic compounds and their use as orexin receptor modulators 詹森药业有限公司 2020-01-10 CN disclosed