SCHEMBL28360807

SCHEMBL28360807

O=C(C=Cc1ccc(O)cc1)C=Cc1ccccn1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F3 P13726 4/20 0.65
CYP2D6 P10635 2/20 0.65
CYP2C9 P11712 2/20 0.65
TYR P14679 2/20 0.65
HSD11B1 P28845 1/20 0.65
HSP90AA1 P07900 1/20 0.53
MAPT P10636 4/20 0.52
ALDH1A1 P00352 2/20 0.52
LMNA P02545 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
PLIN1 O60240 1/20 0.52
CYP1A2 P05177 1/20 0.52
RECQL P46063 1/20 0.52
PLIN5 Q00G26 1/20 0.52
ABHD5 Q8WTS1 1/20 0.52
GSK3B P49841 2/20 0.51
BACE1 P56817 2/20 0.51
TLR9 Q9NR96 1/20 0.51
KMT2A Q03164 4/20 0.50
PKM P14618 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11999794 0.88 MAPT (0.68) F3CYP2D6CYP2C9HSP90AA1MAPT
SCHEMBL3216593 0.88 AKR1B10 (0.67) HSP90AA1GSK3BBACE1AKR1B10AKR1B1
SCHEMBL3216578 0.88 AKR1B10 (0.67) HSP90AA1GSK3BBACE1AKR1B10AKR1B1
Hydrochloric Acid SCHEMBL11971239 0.87 MAPT (0.66) F3CYP2D6CYP2C9HSP90AA1MAPT
Hydrochloric Acid SCHEMBL11971243 0.87 MAPT (0.66) F3CYP2D6CYP2C9HSP90AA1MAPT
SCHEMBL30317323 0.86 NPC1 (0.62) F3CYP2D6CYP2C9HSP90AA1MAPT
SCHEMBL11999774 0.86 NPC1 (0.62) F3CYP2D6CYP2C9HSP90AA1MAPT
SCHEMBL7802342 0.83 KMT2A (0.64) CYP2D6CYP2C9MAPTALDH1A1LMNA
SCHEMBL9605431 0.83 KMT2A (0.64) CYP2D6CYP2C9MAPTALDH1A1LMNA
SCHEMBL10053044 0.81 F3 (0.83) F3CYP2D6CYP2C9TYRHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108530435-B Quinoxaline-containing 1, 4-pentadiene-3-ketone derivative, preparation method and application 贵州大学 2021-08-17 CN disclosed
CN-108822045-B Quinazoline-containing 1, 4-pentadiene-3-ketoxime ether derivative, preparation method and application 贵州大学 2021-06-08 CN disclosed
CN-107056687-B Pyridine group-containing 1, 4-pentadiene-3-ketoxime ester compound, preparation method and application 贵州大学 2020-06-30 CN disclosed
CN-108530427-B Quinazoline-containing 1, 4-pentadiene-3-ketoxime ether derivative, and preparation method and application thereof 贵州大学 2020-05-08 CN disclosed
CN-106928176-B Coumarin-containing 1, 4-pentadiene-3-ketone derivative and preparation method and application thereof 贵州大学 2020-02-18 CN disclosed