SCHEMBL28374191

SCHEMBL28374191

COc1c(OC(C)=O)ccc2c1N=C(C=C(O)c1cccnc1)N1CCN=C21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.36
CYP1A1 P04798 3/20 0.36
CYP1A2 P05177 3/20 0.36
CYP1B1 Q16678 3/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
TDP1 Q9NUW8 1/20 0.35
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
THRB P10828 1/20 0.33
GPR6 P46095 1/20 0.33
PIK3CD O00329 1/20 0.33
PIK3C2A O00443 1/20 0.33
PIK3C2B O00750 1/20 0.33
PIK3R1 P27986 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33
PRKDC P78527 1/20 0.33
PIK3C3 Q8NEB9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL82158 0.91 CYP1A1 (0.39) POLBCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL29475061 0.91 CYP1A1 (0.39) POLBCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL82157 0.91 CYP1A1 (0.39) POLBCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL86657 0.91 CYP1A1 (0.39) POLBCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL82967 0.88 CYP1A1 (0.35) POLBCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL29475036 0.88 CYP1A1 (0.35) POLBCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL82968 0.88 CYP1A1 (0.35) POLBCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL15119595 0.88 TBXAS1 (0.33) POLBCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL86825 0.88 KMT2A (0.36) POLBTDP1ALDH1A1GPR6PIK3CB
SCHEMBL86675 0.87 KMT2A (0.33) POLBCYP1A1CYP1A2CYP1B1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109729716-B PI3K inhibitor combination 拜耳制药股份公司 2022-03-15 CN disclosed
CN-105934256-B PI3K inhibitor combination 拜耳制药股份公司 2019-12-27 CN disclosed