SCHEMBL28374459

SCHEMBL28374459

Cn1cnc(C(C)(N)CC(=O)O)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.35
TSHR P16473 2/20 0.35
CYP2C9 P11712 1/20 0.35
MTOR P42345 1/20 0.35
HRH4 Q9H3N8 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
CPB2 Q96IY4 1/20 0.34
HIF1A Q16665 2/20 0.33
MAPK8 P45983 1/20 0.32
MAPK10 P53779 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HMGCR P04035 1/20 0.31
CHRM1 P11229 1/20 0.31
TBXA2R P21731 1/20 0.31
ADRA1A P35348 1/20 0.31
CYP2D6 P10635 1/20 0.31
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18074293 1.00 CYP2C19 (0.35) CYP2C19TSHRCYP2C9MTORHRH4
SCHEMBL28373091 0.83 MAPK8 (0.37) CYP2C19TSHRCYP2C9MTORHRH4
SCHEMBL1045230 0.74 CYP2C9 (0.36) CYP2C19TSHRCYP2C9MTORHRH4
SCHEMBL8472358 0.73 CYP2C9 (0.39) CYP2C19TSHRCYP2C9MTORHRH4
SCHEMBL18074299 0.71 KDM4E (0.36) CYP2C19TSHRTDP1HIF1AKDM4E
SCHEMBL28368784 0.71 KDM4E (0.36) CYP2C19TSHRTDP1HIF1AKDM4E
SCHEMBL12928753 0.70 CYP2C9 (0.36) CYP2C19TSHRCYP2C9MTORHRH4
SCHEMBL18074340 0.70 CYP2C19 (0.38) CYP2C19TSHRHIF1AKDM4EHMGCR
SCHEMBL18074328 0.70 ALDH1A1 (0.39) CYP2C19HIF1AKDM4EALDH1A1
SCHEMBL25015250 0.70 CYP2C9 (0.38) CYP2C19TSHRCYP2C9MTORHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107207481-B 3- (4-ethynylphenyl) hexahydropyrimidine-2, 4-dione derivatives as modulators of MGLUR4 豪夫迈·罗氏有限公司 2020-03-03 CN disclosed