SCHEMBL28378952

SCHEMBL28378952

COC(=O)C1(CO[Si](C)(C)C(C)(C)C)CCN(Cc2ccccc2)C1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 6/20 0.47
ALDH1A1 P00352 1/20 0.47
KDM4E B2RXH2 1/20 0.45
GAA P10253 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
POLB P06746 1/20 0.43
CYP3A4 P08684 3/20 0.43
TSHR P16473 3/20 0.43
LMNA P02545 1/20 0.42
KCNH2 Q12809 4/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2467441 0.91 KDM4E (0.56) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL2470923 0.85 CYP2D6 (0.54) CYP2D6ALDH1A1KDM4EGAAMEN1
SCHEMBL19779408 0.81 KMT2A (0.53) CYP2D6ALDH1A1KDM4EGAAMEN1
SCHEMBL1961694 0.80 KMT2A (0.52) CYP2D6ALDH1A1KDM4EGAAMEN1
SCHEMBL15367649 0.79 KMT2A (0.53) CYP2D6ALDH1A1KDM4EGAAMEN1
SCHEMBL14517088 0.79 CYP2D6 (0.50) CYP2D6ALDH1A1KDM4EGAAMEN1
SCHEMBL4299006 0.79 NPFFR1 (0.51) CYP2D6ALDH1A1KMT2AL3MBTL1CYP3A4
SCHEMBL2468808 0.78 CYP2D6 (0.49) CYP2D6ALDH1A1KDM4EGAAMEN1
SCHEMBL2470540 0.78 CYP2D6 (0.47) CYP2D6ALDH1A1KDM4EGAAMEN1
SCHEMBL18203100 0.76 L3MBTL1 (0.63) CYP2D6ALDH1A1GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105732636-B Heteroaromatic compounds and their use in medicine 广东东阳光药业有限公司 2020-04-21 CN disclosed