SCHEMBL28385331

SCHEMBL28385331

OC1CC2(CCNC2)Oc2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 7/20 0.55
KCNH2 Q12809 7/20 0.43
CYP2D6 P10635 3/20 0.43
SCD O00767 1/20 0.36
KMT2A Q03164 1/20 0.35
HDAC3 O15379 2/20 0.34
HDAC4 P56524 2/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC7 Q8WUI4 2/20 0.34
HDAC2 Q92769 2/20 0.34
HDAC10 Q969S8 2/20 0.34
HDAC11 Q96DB2 2/20 0.34
HDAC8 Q9BY41 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
HDAC9 Q9UKV0 2/20 0.34
HDAC5 Q9UQL6 2/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
HTR2A P28223 1/20 0.33
MAOA P21397 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12481110 0.91 OPRD1 (0.65) OPRD1KCNH2CYP2D6SCDKMT2A
SCHEMBL30538347 0.91 OPRD1 (0.65) OPRD1KCNH2CYP2D6SCDKMT2A
SCHEMBL20109488 0.88 OPRD1 (0.46) OPRD1KCNH2CYP2D6SCDKMT2A
SCHEMBL11244376 0.80 OPRD1 (0.47) OPRD1KCNH2CYP2D6SCDKMT2A
SCHEMBL15717425 0.80 OPRD1 (0.47) OPRD1KCNH2CYP2D6SCDKMT2A
SCHEMBL1115144 0.78 OPRD1 (0.46) OPRD1KCNH2CYP2D6SCDKMT2A
SCHEMBL12162414 0.78 OPRD1 (0.46) OPRD1KCNH2CYP2D6SCDKMT2A
SCHEMBL5312276 0.73 KMT2A (0.62) OPRD1SCDKMT2AHDAC3HDAC4
SCHEMBL16503896 0.73 KMT2A (0.46) OPRD1KCNH2CYP2D6SCDKMT2A
SCHEMBL12481437 0.73 OPRD1 (0.62) OPRD1KCNH2CYP2D6KMT2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111094293-A Substituted benzoxazole and benzofuran compounds as PDE7 inhibitors 达特神经科学有限公司 2020-05-01 CN claimed
CN-111094293-A Substituted benzoxazole and benzofuran compounds as PDE7 inhibitors 达特神经科学有限公司 2020-05-01 CN disclosed