SCHEMBL28392011

SCHEMBL28392011

COc1cc(OC(N)=O)c(N)cc1C(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.46
CYP3A4 P08684 2/20 0.46
TP53 P04637 1/20 0.46
HPGD P15428 1/20 0.46
ALOX15 P16050 1/20 0.46
HTR2A P28223 1/20 0.41
ALDH1A1 P00352 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
HTT P42858 1/20 0.40
RARA P10276 2/20 0.38
RARB P10826 2/20 0.38
RARG P13631 2/20 0.38
GAA P10253 2/20 0.37
KDM4E B2RXH2 1/20 0.37
PKM P14618 1/20 0.37
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28388909 0.78 GAA (0.35) ALDH1A1GAAKDM4EPTGDR2NR1H4
SCHEMBL1421221 0.78 ALDH1A1 (0.46) LMNACYP3A4TP53HPGDALOX15
SCHEMBL28532035 0.74 KDM4E (0.39) ALOX15ALDH1A1L3MBTL1HTTRARA
SCHEMBL15422590 0.73 NR1H4 (0.42) LMNAALOX15ALDH1A1RARARARB
SCHEMBL28392012 0.73 CA1 (0.47) LMNACYP3A4TP53HPGDALOX15
SCHEMBL92809 0.72 CYP3A4 (0.64) LMNACYP3A4TP53HPGDALOX15
SCHEMBL28526640 0.72 KDM4E (0.45) HPGDALOX15ALDH1A1L3MBTL1HTT
SCHEMBL19393881 0.71 CYP3A4 (0.53) LMNACYP3A4TP53HPGDALOX15
SCHEMBL12781654 0.70 CYP3A4 (0.68) LMNACYP3A4TP53HPGDALOX15
SCHEMBL16767200 0.70 ALDH1A1 (0.50) LMNAHPGDALOX15ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111116469-A HDAC inhibitor, preparation method, pharmaceutical composition and application thereof 北京鑫开元医药科技有限公司 2020-05-08 CN disclosed