SCHEMBL28404707

SCHEMBL28404707

CC(NC(=O)c1cc(N)ccc1N(C)C)c1cccc2ccccc12

nearest known ligand 0.75

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
LMNA P02545 1/20 0.51
GAA P10253 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29494539 1.00 MEN1 (0.53) MEN1KMT2ALMNAGAA
SCHEMBL29793667 1.00 MEN1 (0.53) MEN1KMT2ALMNAGAA
SCHEMBL27382820 0.86 ALOX5 (0.59) MEN1KMT2ALMNAGAA
SCHEMBL30344651 0.86
SCHEMBL27382823 0.86 ALOX5 (0.59) MEN1KMT2ALMNAGAA
SCHEMBL1319181 0.86
SCHEMBL29494494 0.86
SCHEMBL29449377 0.86
SCHEMBL21067703 0.86
SCHEMBL30966415 0.85 MEN1 (0.54) MEN1KMT2ALMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108929263-B Arylamide Kv2.1 inhibitor and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-07-22 CN disclosed
CN-111108092-A Arylamide Kv2.1 inhibitor and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2020-05-05 CN disclosed