SCHEMBL28404709

SCHEMBL28404709

[CH2]Cc1cccc(C(C)N)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 9/20 0.37
HRH4 Q9H3N8 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
SLC6A2 P23975 2/20 0.32
TAAR1 Q96RJ0 2/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
MAOA P21397 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
CYP2A6 P11509 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29337105 0.81 IRAK4 (0.44) IRAK4
SCHEMBL2936127 0.81 IRAK4 (0.44) IRAK4
SCHEMBL21455525 0.80 IRAK4 (0.38) IRAK4
SCHEMBL522063 0.79 CYP1A2 (0.38) IRAK4SLC6A2TAAR1MAOASLC6A4
SCHEMBL25170530 0.75 NOS3 (0.48) IRAK4NOS2
SCHEMBL29793597 0.75 NOS3 (0.48) IRAK4NOS2
SCHEMBL18793683 0.75 NOS3 (0.48) IRAK4NOS2
SCHEMBL1509600 0.75 NOS3 (0.48) IRAK4NOS2
SCHEMBL2364924 0.75 KCNH2 (0.62) NOS1NOS2
SCHEMBL1515200 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111108092-A Arylamide Kv2.1 inhibitor and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2020-05-05 CN disclosed