SCHEMBL28405182

SCHEMBL28405182

O=C(O)Cn1cc(-c2cccc(NC(=O)c3ccccc3F)c2)nn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.54
HSD17B10 Q99714 1/20 0.54
TP53 P04637 2/20 0.53
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
LCLAT1 Q6UWP7 2/20 0.51
MAPT P10636 1/20 0.51
UCHL5 Q9Y5K5 1/20 0.49
SIRT2 Q8IXJ6 1/20 0.49
HDAC3 O15379 3/20 0.48
HDAC1 Q13547 3/20 0.48
HDAC2 Q92769 3/20 0.48
HDAC10 Q969S8 3/20 0.48
HDAC8 Q9BY41 3/20 0.48
HDAC6 Q9UBN7 3/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
RGS12 O14924 1/20 0.48
PABPC1 P11940 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29863008 1.00 KDM4E (0.54) KDM4EHSD17B10TP53MEN1KMT2A
SCHEMBL29863433 0.84 MEN1 (0.51) MEN1KMT2ASMN1; SMN2MAPTUCHL5
SCHEMBL28405517 0.84 MEN1 (0.51) MEN1KMT2ASMN1; SMN2MAPTUCHL5
SCHEMBL28401956 0.83 TP53 (0.53) KDM4ETP53MEN1KMT2ASMN1; SMN2
SCHEMBL29862961 0.83 TP53 (0.53) KDM4ETP53MEN1KMT2ASMN1; SMN2
SCHEMBL29862908 0.81 HDAC3 (0.54) KDM4EHSD17B10TP53MEN1KMT2A
SCHEMBL28400450 0.81 HDAC3 (0.54) KDM4EHSD17B10TP53MEN1KMT2A
SCHEMBL28398052 0.81 AURKA (0.48) UCHL5SIRT2HDAC3HDAC1HDAC2
SCHEMBL29863097 0.81 AURKA (0.48) UCHL5SIRT2HDAC3HDAC1HDAC2
SCHEMBL28397320 0.80 TP53 (0.52) KDM4EHSD17B10TP53MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111057015-A 2- (4-phenyl-1H-1, 2, 3-triazole-1-yl) acetic acid and acethydrazide compounds 中国医科大学 2020-04-24 CN claimed
CN-111057015-B 2- (4-phenyl-1H-1, 2, 3-triazole-1-yl) acetic acid and acethydrazide compounds 中国医科大学 2022-09-16 CN disclosed
CN-111057015-A 2- (4-phenyl-1H-1, 2, 3-triazole-1-yl) acetic acid and acethydrazide compounds 中国医科大学 2020-04-24 CN disclosed