SCHEMBL29863433

SCHEMBL29863433

O=C(O)Cn1cc(-c2cccc(NC(=O)c3ccccc3[N+](=O)[O-])c2)nn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
HTT P42858 2/20 0.47
UCHL5 Q9Y5K5 1/20 0.47
GAA P10253 1/20 0.47
NCOA1 Q15788 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NCOA3 Q9Y6Q9 1/20 0.47
SIRT2 Q8IXJ6 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.46
HDAC3 O15379 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC10 Q969S8 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
ALOX5 P09917 1/20 0.46
PTGES2 Q9H7Z7 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28405517 1.00 MEN1 (0.51) MEN1KMT2AHTTUCHL5GAA
SCHEMBL29863008 0.84 KDM4E (0.54) MEN1KMT2AHTTUCHL5GAA
SCHEMBL28405182 0.84 KDM4E (0.54) MEN1KMT2AHTTUCHL5GAA
SCHEMBL29862908 0.78 HDAC3 (0.54) MEN1KMT2AUCHL5SMN1; SMN2SIRT2
SCHEMBL28400450 0.78 HDAC3 (0.54) MEN1KMT2AUCHL5SMN1; SMN2SIRT2
SCHEMBL28398052 0.78 AURKA (0.48) HTTUCHL5SIRT2HDAC3HDAC1
SCHEMBL29863097 0.78 AURKA (0.48) HTTUCHL5SIRT2HDAC3HDAC1
SCHEMBL29863344 0.77 TP53 (0.52) MEN1KMT2AUCHL5SMN1; SMN2HDAC3
SCHEMBL28397320 0.77 TP53 (0.52) MEN1KMT2AUCHL5SMN1; SMN2HDAC3
SCHEMBL29862961 0.76 TP53 (0.53) MEN1KMT2ASMN1; SMN2HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111057015-B 2- (4-phenyl-1H-1, 2, 3-triazole-1-yl) acetic acid and acethydrazide compounds 中国医科大学 2022-09-16 CN disclosed