SCHEMBL28406503

SCHEMBL28406503

CC(C)(C)OC(=O)NCCCCC(NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N1CCC(C(=O)ONC(=O)OCc2ccccc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.55
ITGA2B P08514 1/20 0.55
TGM2 P21980 14/20 0.50
F13A1 P00488 2/20 0.50
TGM1 P22735 2/20 0.50
TGM6 O95932 1/20 0.47
TLR2 O60603 1/20 0.46
TLR1 Q15399 1/20 0.46
KLK7 P49862 1/20 0.45
KLK5 Q9Y337 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28447032 0.91 ITGB3 (0.62) ITGB3ITGA2BTGM2F13A1TGM1
SCHEMBL13702142 0.85 TLR2 (0.53) ITGB3ITGA2BTGM2F13A1TGM1
SCHEMBL21009949 0.85 ITGB3 (0.52) ITGB3ITGA2BTGM2F13A1TGM1
SCHEMBL29930528 0.85 ITGB3 (0.52) ITGB3ITGA2BTGM2F13A1TGM1
SCHEMBL19708135 0.85 ITGB3 (0.52) ITGB3ITGA2BTGM2F13A1TGM1
SCHEMBL22694079 0.85 ITGB3 (0.51) ITGB3ITGA2BTGM2F13A1TGM1
SCHEMBL20975607 0.84 ITGB3 (0.52) ITGB3ITGA2BTGM2F13A1TGM1
SCHEMBL28399421 0.83 DPP7 (0.57) ITGB3ITGA2BTGM2F13A1TGM1
SCHEMBL22582335 0.83 ITGB3 (0.49) ITGB3ITGA2BTGM2F13A1TGM1
SCHEMBL14064950 0.82 KLK7 (0.54) ITGB3ITGA2BTLR2TLR1KLK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111065390-B Use of a KOR agonist in combination with a MOR agonist for the preparation of a medicament for the treatment of pain 江苏恒瑞医药股份有限公司 2023-01-24 CN disclosed
CN-114940700-A Phenyl propionamide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-08-26 CN disclosed
CN-108290926-B Phenyl propionamide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-02-08 CN disclosed
CN-111065631-B Salt of phenylpropionamide derivative and preparation method thereof 江苏恒瑞医药股份有限公司 2021-10-08 CN disclosed
CN-109879934-B Salt of phenylpropionamide derivative and preparation method thereof 江苏恒瑞医药股份有限公司 2020-12-08 CN disclosed
CN-111065390-A Use of a KOR agonist in combination with a MOR agonist for the preparation of a medicament for the treatment of pain 江苏恒瑞医药股份有限公司 2020-04-24 CN disclosed
CN-111065631-A Salt of phenylpropionamide derivative and preparation method thereof 江苏恒瑞医药股份有限公司 2020-04-24 CN disclosed