SCHEMBL28407299

SCHEMBL28407299

CC(C)(C)NC(=O)O[C@@H](C(=O)NC1CC1)C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.37
HDAC4 P56524 3/20 0.36
HDAC1 Q13547 3/20 0.36
HPGD P15428 2/20 0.33
TSHR P16473 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GAA P10253 2/20 0.33
HTT P42858 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
EPHX1 P07099 1/20 0.33
HDAC6 Q9UBN7 1/20 0.32
SMYD3 Q9H7B4 1/20 0.32
EPHX2 P34913 1/20 0.32
PKM P14618 1/20 0.32
MAPT P10636 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28407625 0.80 SMYD3 (0.36) KMT2AHPGDTSHRNPSR1HTT
SCHEMBL28407622 0.80 SMYD3 (0.36) KMT2AHPGDTSHRNPSR1HTT
SCHEMBL28889722 0.78 SCN9A (0.32)
SCHEMBL27823739 0.76 HIF1A (0.32)
SCHEMBL28854942 0.75 HPGD (0.49) KMT2AHDAC4HDAC1HPGDTSHR
SCHEMBL14283011 0.73 POLB (0.32) KMT2AGAA
SCHEMBL8261900 0.73 POLB (0.32) KMT2AGAA
SCHEMBL28737429 0.73 EPHX1 (0.42) KMT2AHDAC4HDAC1HPGDGAA
SCHEMBL28038198 0.71 HDAC4 (0.34) KMT2AHDAC4HDAC1HPGDGAA
SCHEMBL3216743 0.69 POLB (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111225900-A 3, 4-disubstituted 3-cyclobutene-1, 2-diones and their use 阿勒根公司 2020-06-02 CN disclosed