SCHEMBL28408693

SCHEMBL28408693

CC(=O)N1C(=O)C(=C(O)c2ccc(Cl)cc2)c2cc([N+](=O)[O-])ccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
LMNA P02545 3/20 0.44
SNCA P37840 3/20 0.44
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
KDM4E B2RXH2 2/20 0.42
NPC1 O15118 2/20 0.42
HTT P42858 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
CASP1 P29466 2/20 0.41
CASP3 P42574 2/20 0.41
CASP4 P49662 2/20 0.41
CASP7 P55210 2/20 0.41
CASP9 P55211 2/20 0.41
CASP6 P55212 2/20 0.41
CASP8 Q14790 1/20 0.41
MAPT P10636 4/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8009607 0.90 CA12 (0.46) ALDH1A1LMNASNCACA12CA9
SCHEMBL8009610 0.90 CA12 (0.46) ALDH1A1LMNASNCACA12CA9
SCHEMBL6328682 0.89 ALDH1A1 (0.44) ALDH1A1LMNASNCACA12CA9
SCHEMBL6328679 0.89 ALDH1A1 (0.44) ALDH1A1LMNASNCACA12CA9
SCHEMBL8010164 0.89 MEN1 (0.44) ALDH1A1LMNASNCACA12CA9
SCHEMBL8010160 0.89 MEN1 (0.44) ALDH1A1LMNASNCACA12CA9
SCHEMBL4480293 0.87 CES1 (0.41) ALDH1A1LMNASNCACA12CA9
SCHEMBL4480297 0.87 CES1 (0.41) ALDH1A1LMNASNCACA12CA9
SCHEMBL4300695 0.86 MAPK1 (0.48) ALDH1A1LMNASNCACA12CA9
SCHEMBL4300692 0.86 MAPK1 (0.48) ALDH1A1LMNASNCACA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111285872-B Indole-2-ketone derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2022-05-17 CN disclosed
CN-111285872-A Indole-2-ketone derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2020-06-16 CN disclosed