SCHEMBL28409102

SCHEMBL28409102

COC1(C(=O)O)CC=C(c2nc(Nc3cc(C)[nH]n3)c3ccccc3n2)CC1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AURKA O14965 15/20 0.55
AURKB Q96GD4 12/20 0.55
GSK3B P49841 8/20 0.55
SRC P12931 6/20 0.55
EIF2AK2 P19525 1/20 0.55
GSK3A P49840 1/20 0.55
JAK2 O60674 3/20 0.46
CYP3A4 P08684 3/20 0.46
CYP2C8 P10632 3/20 0.46
CYP2C9 P11712 3/20 0.46
JAK1 P23458 3/20 0.46
TYK2 P29597 3/20 0.46
CYP2C19 P33261 3/20 0.46
JAK3 P52333 3/20 0.46
ADORA3 P0DMS8 2/20 0.46
CYP1A2 P05177 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30250187 0.94 AURKA (0.54) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL24668009 0.94 AURKA (0.54) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL28415530 0.87 AURKA (0.40) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL30250065 0.87 AURKA (0.40) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL30249999 0.86 PAK1 (0.45) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL30249931 0.86 AURKA (0.39) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL30250129 0.80 AURKA (0.38) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL28416436 0.80 AURKA (0.38) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL28411553 0.79 RET (0.61) JAK2
SCHEMBL30250189 0.79 PAK1 (0.45) AURKAAURKBGSK3BSRCEIF2AK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111285882-B Fused ring compound, pharmaceutical composition containing same, and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2022-12-02 CN disclosed
CN-111285882-A Fused ring compound, pharmaceutical composition containing same, and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2020-06-16 CN disclosed