SCHEMBL30250065

SCHEMBL30250065

COC1(C(=O)O)CC=C(c2nc(Nc3cc(C)[nH]n3)c3cc[nH]c3n2)CC1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AURKA O14965 12/20 0.40
AURKB Q96GD4 8/20 0.40
SRC P12931 2/20 0.39
GSK3B P49841 2/20 0.39
EIF2AK2 P19525 1/20 0.39
GSK3A P49840 1/20 0.39
PAK4 O96013 4/20 0.37
RET P07949 1/20 0.37
TGFBR1 P36897 2/20 0.36
TGFBR2 P37173 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28415530 1.00 AURKA (0.40) AURKAAURKBSRCGSK3BEIF2AK2
SCHEMBL28416436 0.93 AURKA (0.38) AURKAAURKBSRCGSK3BEIF2AK2
SCHEMBL30250129 0.93 AURKA (0.38) AURKAAURKBSRCGSK3BEIF2AK2
SCHEMBL28409102 0.87 AURKA (0.55) AURKAAURKBSRCGSK3BEIF2AK2
SCHEMBL30249931 0.85 AURKA (0.39) AURKAAURKBSRCGSK3BEIF2AK2
SCHEMBL30249999 0.82 PAK1 (0.45) AURKAAURKBSRCGSK3BEIF2AK2
SCHEMBL24668009 0.81 AURKA (0.54) AURKAAURKBSRCGSK3BEIF2AK2
SCHEMBL30250187 0.81 AURKA (0.54) AURKAAURKBSRCGSK3BEIF2AK2
SCHEMBL28411559 0.78 RET (0.44) AURKAAURKBSRCGSK3BPAK4
SCHEMBL30250267 0.78 RET (0.44) AURKAAURKBSRCGSK3BPAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111285882-B Fused ring compound, pharmaceutical composition containing same, and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2022-12-02 CN disclosed