SCHEMBL28413504

SCHEMBL28413504

CC(NC(=O)c1cc(N)ccc1N(C)C)c1cccc(-c2ccco2)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNB1 Q14721 1/20 0.45
KCNB2 Q92953 1/20 0.45
TP53 P04637 1/20 0.39
KDM4E B2RXH2 2/20 0.39
TSHR P16473 1/20 0.39
RECQL P46063 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KEAP1 Q14145 1/20 0.38
ALOX5 P09917 1/20 0.37
BLK P51451 1/20 0.36
BTK Q06187 1/20 0.36
PSMB5 P28074 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29793721 1.00 KCNB1 (0.45) KCNB1KCNB2TP53KDM4ETSHR
SCHEMBL28406253 0.85 KCNB1 (0.56) KCNB1KCNB2KDM4EHSD17B10ALDH1A1
SCHEMBL28410953 0.84 KCNB1 (0.68) KCNB1KCNB2KDM4EALDH1A1
SCHEMBL28406352 0.84 MAPT (0.48) KCNB1KCNB2TP53KDM4ETSHR
SCHEMBL29793887 0.80 KCNB1 (0.66) KCNB1KCNB2KDM4EHSD17B10ALDH1A1
SCHEMBL28257362 0.80 KCNB1 (0.66) KCNB1KCNB2KDM4EHSD17B10ALDH1A1
SCHEMBL29793613 0.80 KCNB1 (0.51) KCNB1KDM4EHSD17B10ALDH1A1PSMB5
SCHEMBL28409921 0.80 KCNB1 (0.51) KCNB1KDM4EHSD17B10ALDH1A1PSMB5
SCHEMBL29793727 0.78 KCNB1 (0.55) KCNB1KCNB2
SCHEMBL28257384 0.78 KCNB1 (0.55) KCNB1KCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108929263-B Arylamide Kv2.1 inhibitor and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-07-22 CN disclosed
CN-111108092-A Arylamide Kv2.1 inhibitor and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2020-05-05 CN disclosed