SCHEMBL2841353

SCHEMBL2841353

N#Cc1ccccc1N1CCN(C(=O)C2CC(NCc3ccc(Cl)c(Cl)c3)CN2Cc2ccccc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.42
CHRM4 P08173 3/20 0.41
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
RECQL P46063 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MC4R P32245 1/20 0.40
DPP4 P27487 1/20 0.39
KDM1A O60341 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
DRD2 P14416 2/20 0.39
DRD4 P21917 2/20 0.39
DRD3 P35462 1/20 0.39
GRM5 P41594 1/20 0.39
NPBWR1 P48145 1/20 0.39
MCHR1 Q99705 1/20 0.39
P2RY12 Q9H244 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2817861 1.00 TACR1 (0.42) TACR1CHRM4MEN1LMNAHTT
SCHEMBL2817089 0.93 DPP4 (0.43) CHRM4MC4RDPP4KDM1AMAOA
SCHEMBL13841884 0.92 DRD2 (0.44) CHRM4MC4RDPP4DRD2DRD4
SCHEMBL2821338 0.92 DRD2 (0.44) CHRM4MC4RDPP4DRD2DRD4
SCHEMBL2821782 0.91 DPP4 (0.45) CHRM4MC4RDPP4KDM1ADRD2
SCHEMBL2817914 0.91 DRD2 (0.47) CHRM4LMNAMC4RDPP4KDM1A
SCHEMBL2822155 0.90 CHRM4 (0.44) CHRM4MC4RDPP4DRD2DRD4
SCHEMBL2818985 0.88 NPFFR1 (0.42) CHRM4HTTMC4RDPP4DRD2
SCHEMBL2839427 0.88 BCHE (0.46) CHRM4MC4RDPP4DRD2DRD4
SCHEMBL2839423 0.88 BCHE (0.46) CHRM4MC4RDPP4DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155672-B1 PROLINAMIDE DERIVATIVES AS NK3 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-10-27 EP disclosed