SCHEMBL28414844

SCHEMBL28414844

CCS(=O)(=O)NC1C(=O)Nc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 6/20 0.43
MAPT P10636 5/20 0.43
ALDH1A1 P00352 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
TDO2 P48775 2/20 0.42
KDM4E B2RXH2 4/20 0.41
NLRP3 Q96P20 1/20 0.41
GAA P10253 1/20 0.40
GSK3B P49841 1/20 0.39
HPGDS O60760 1/20 0.38
BRPF1 P55201 1/20 0.38
CREBBP Q92793 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24754644 0.76 IDO1 (0.46) IDO1MAPTALDH1A1L3MBTL1TDO2
SCHEMBL28827997 0.73 IDO1 (0.44) IDO1MAPTALDH1A1L3MBTL1TDO2
SCHEMBL1491212 0.73 KDM4E (0.47) IDO1MAPTALDH1A1L3MBTL1TDO2
SCHEMBL28859743 0.73 IDO1 (0.46) IDO1MAPTALDH1A1L3MBTL1TDO2
SCHEMBL29197967 0.73 IDO1 (0.50) IDO1MAPTALDH1A1L3MBTL1TDO2
SCHEMBL10338752 0.73 KDM4E (0.57) IDO1MAPTALDH1A1L3MBTL1TDO2
SCHEMBL8226202 0.72 MAPT (0.43) IDO1MAPTALDH1A1L3MBTL1TDO2
Hydrochloric Acid SCHEMBL1491278 0.72 KDM4E (0.46) IDO1MAPTALDH1A1L3MBTL1TDO2
SCHEMBL2693278 0.69 IDO1 (0.64) IDO1MAPTALDH1A1L3MBTL1TDO2
SCHEMBL19000599 0.69 IDO1 (0.51) IDO1MAPTALDH1A1L3MBTL1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111285872-B Indole-2-ketone derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2022-05-17 CN disclosed
CN-111285872-A Indole-2-ketone derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2020-06-16 CN disclosed