SCHEMBL28419174

SCHEMBL28419174

CCOC(=O)c1nccn1CCCN(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
PKM P14618 1/20 0.40
CYP2C19 P33261 1/20 0.40
ALDH1A1 P00352 5/20 0.39
KMT2A Q03164 4/20 0.39
POLB P06746 2/20 0.39
HPGD P15428 3/20 0.37
JMJD6 Q6NYC1 1/20 0.37
TBXAS1 P24557 1/20 0.37
RGS12 O14924 1/20 0.37
MAPT P10636 1/20 0.37
KDM5A P29375 1/20 0.36
KDM5C P41229 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
KDM4E B2RXH2 2/20 0.36
HSD17B10 Q99714 1/20 0.36
RAD52 P43351 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28420055 0.92 SMN1; SMN2 (0.40) CYP1A2CYP3A4CYP2C9PKMCYP2C19
SCHEMBL27486503 0.86 ALDH1A1 (0.54) CYP1A2CYP3A4CYP2C9PKMCYP2C19
SCHEMBL4118014 0.83 ALDH1A1 (0.41) CYP1A2CYP3A4CYP2C9PKMCYP2C19
SCHEMBL30554011 0.83 ALDH1A1 (0.41) CYP1A2CYP3A4CYP2C9PKMCYP2C19
SCHEMBL30554028 0.83 JMJD6 (0.42) CYP1A2CYP3A4CYP2C9PKMCYP2C19
SCHEMBL1838525 0.82 TNF (0.47)
SCHEMBL28413273 0.81 SMN1; SMN2 (0.40) CYP1A2CYP3A4CYP2C9PKMCYP2C19
SCHEMBL1422820 0.81 CYP1A2 (0.45) CYP1A2CYP3A4CYP2C9PKMCYP2C19
SCHEMBL30554005 0.80 JMJD6 (0.40) CYP1A2ALDH1A1KMT2AHPGDJMJD6
SCHEMBL30554008 0.80 JMJD6 (0.40) CYP1A2ALDH1A1KMT2APOLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111187218-B Application of 1-substituted-1H-imidazole-2-carboxylic acid compound in preparation of metal beta-lactamase inhibitor 四川大学 2023-08-04 CN disclosed
CN-111253317-B 1-substituted-1H-imidazole-2-carboxylic acid compound 四川大学 2023-08-04 CN disclosed
CN-111253317-A 1-substituted-1H-imidazole-2-carboxylic acid compound 四川大学 2020-06-09 CN disclosed
CN-111187218-A Application of 1-substituted-1H-imidazole-2-carboxylic acid compounds in preparation of metal β -lactamase inhibitor 四川大学 2020-05-22 CN disclosed