SCHEMBL28420161

SCHEMBL28420161

CCCSc1cc(C(=O)NN)ccn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.45
MPO P05164 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2A6 P11509 1/20 0.45
CYP2C19 P33261 1/20 0.45
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
HPGD P15428 1/20 0.44
HTT P42858 1/20 0.42
ALDH1A1 P00352 3/20 0.38
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
TP53 P04637 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28851024 0.88 KDM4E (0.47) KDM4EMPOCYP1A2CYP3A4ADORA3
SCHEMBL29123005 0.85 DDB1 (0.43) KDM4ECYP1A2CYP3A4NPC1RAB9A
SCHEMBL2998832 0.74 KDM4E (0.64) KDM4EMPOCYP1A2CYP3A4ADORA3
SCHEMBL2989555 0.73 CYP1A2 (0.60) KDM4EMPOCYP1A2CYP3A4ADORA3
SCHEMBL10796248 0.73 DDB1 (0.46) KDM4ECYP1A2CYP3A4NPC1RAB9A
SCHEMBL1543956 0.73 KDM4E (0.55) KDM4EMPOCYP1A2CYP3A4ADORA3
SCHEMBL30637340 0.73 KDM4E (0.55) KDM4EMPOCYP1A2CYP3A4ADORA3
SCHEMBL2993048 0.71 KDM4E (0.49) KDM4EMPOCYP1A2CYP3A4ADORA3
SCHEMBL11155559 0.71 KDM4E (0.49) KDM4EMPOCYP1A2CYP3A4ADORA3
SCHEMBL1417739 0.71 GABRP (0.63) KDM4EMPOCYP1A2CYP3A4ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115629139-A Method for determining content of impurities in propylthioisoniazid by using HPLC (high performance liquid chromatography) 江苏慈星药业有限公司 2023-01-20 CN claimed
CN-115616113-A Method for determining impurity content in clozapine raw material medicine by using HPLC 江苏慈星药业有限公司 2023-01-17 CN claimed
CN-215232183-U A device that is used for propylthio isoniazid amine crude aftertreatment 江苏慈星药业有限公司 2021-12-21 CN claimed
CN-117597138-A Pharmaceutical compositions comprising micrococcum compounds and methods of preparing micrococcum compounds A&J科学有限公司 2024-02-23 CN disclosed
CN-113267584-B HPLC related substance analysis method for medicinal substance 北京亚宝生物药业有限公司 2023-03-17 CN disclosed
CN-113358792-B HPLC content analysis method of medicinal substance 北京亚宝生物药业有限公司 2023-02-24 CN disclosed
CN-115629139-A Method for determining content of impurities in propylthioisoniazid by using HPLC (high performance liquid chromatography) 江苏慈星药业有限公司 2023-01-20 CN disclosed
CN-115629139-A Method for determining content of impurities in propylthioisoniazid by using HPLC (high performance liquid chromatography) 江苏慈星药业有限公司 2023-01-20 CN disclosed
CN-115629139-A Method for determining content of impurities in propylthioisoniazid by using HPLC (high performance liquid chromatography) 江苏慈星药业有限公司 2023-01-20 CN disclosed
CN-114981265-A Compound (I) CTXT私人有限公司 2022-08-30 CN disclosed
CN-113975274-A Cyclofused thiazoline 2-pyridones, method for the production thereof and use thereof for treating and/or preventing tuberculosis 快尔生物技术公司 2022-01-28 CN disclosed
CN-109069492-B Cyclofused thiazoline 2-pyridones, method for the production thereof and use thereof for treating and/or preventing tuberculosis 快尔生物技术公司 2021-12-10 CN disclosed
CN-113380362-A Chronic disease supervision method, platform, system, electronic equipment and storage medium 安徽科大讯飞医疗信息技术有限公司 2021-09-10 CN disclosed
CN-113358792-A HPLC content analysis method of medicinal substance 北京亚宝生物药业有限公司 2021-09-07 CN disclosed
CN-113267584-A HPLC related substance analysis method for medicinal substance 北京亚宝生物药业有限公司 2021-08-17 CN disclosed
CN-111675635-A Compounds and methods for treating infections 尼奥酷里私人有限公司 2020-09-18 CN disclosed
CN-111630036-A Oxoacridinylacetic acid derivatives and methods of use thereof 西利康斯瓦特股份有限公司 2020-09-04 CN disclosed
CN-111246848-A Cyclofused thiazolo 2-pyridones in combination with antitubercular agents 快尔生物技术公司 2020-06-05 CN disclosed