Piperazine

Piperazine

SCHEMBL2842298

C1CNCCN1.CCCC

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ESR1

The experimentally established mechanism targets of Piperazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.55
MAPT P10636 1/20 0.55
PDE4A P27815 1/20 0.55
KDR P35968 1/20 0.55
CXCR4 P61073 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALDH1A1 P00352 1/20 0.33
GNAI3 P08754 4/20 0.32
GNAO1 P09471 4/20 0.32
GNAI1 P63096 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Butane SCHEMBL4155411 0.95 HIF1A (0.46) HIF1AMAPTPDE4AKDRCXCR4
Butane SCHEMBL22619597 0.89 CXCR4 (0.64) HIF1AMAPTPDE4AKDRCXCR4
Propane SCHEMBL3971658 0.86 HIF1A (0.60) HIF1AMAPTPDE4AKDRCXCR4
Piperazine SCHEMBL27557138 0.86
Pyrrolidine SCHEMBL631271 0.84
Piperazine SCHEMBL27708668 0.84 TSHR (0.50) HIF1AMAPTPDE4AKDRCXCR4
Piperazine SCHEMBL27853221 0.82 HIF1A (0.55) HIF1AMAPTPDE4AKDRCXCR4
Azetidine SCHEMBL28080407 0.82
Nonane SCHEMBL10873465 0.81 TSHR (0.57) HIF1AMAPTPDE4AKDRALDH1A1
Piperazine SCHEMBL3344476 0.81 HIF1A (0.43) HIF1AMAPTPDE4AKDRCXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 148 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120136781-A ROR 1-targeted inhibitor and synthesis method and application thereof 北京大学 2025-06-13 CN claimed
CN-118914314-B Quantitative determination method for metastable iron oxide vacancy defect concentration 华中农业大学 2025-05-06 CN claimed
CN-119736013-A Partially crystallized outer coating for marine optical fiber and preparation method thereof 长飞光纤光缆股份有限公司 2025-04-01 CN claimed
CN-119121438-A Anti-gelling spinning method for liquid crystal elastomer fiber 华南理工大学 2024-12-13 CN claimed
CN-118914314-A Quantitative determination method for metastable iron oxide vacancy defect concentration 华中农业大学 2024-11-08 CN claimed
CN-115044206-B Low-loss preparation method of polyimide foam filled honeycomb 江苏中科聚合新材料产业技术研究院有限公司 2024-03-15 CN claimed
CN-112771056-B Metal organic framework phase and crystallite shape control 加利福尼亚大学董事会 2024-02-23 CN claimed
CN-113527681-B Organic silicon doped polyimide soft foam material, and preparation method and application thereof 常州福隆科技新材料有限公司 2023-08-22 CN claimed
CN-112979905-B Block polyurethane polymer, polymer modified bentonite admixture thereof, and preparation and application thereof 江苏苏博特新材料股份有限公司 2023-03-14 CN claimed
CN-115011222-A Single-component polyurea matte seam beautifying agent 安徽硕阳新材料科技有限公司 2022-09-06 CN claimed
CN-103541281-A Railroad sleeper with multiplayer structure ZHAO WEI 2014-01-29 CN claimed
CN-103012712-A Method for preparing organic and inorganic hybridization modified polyurethane chemical grouting material HEBEI TONGCHENG TECHNOLOGY CO LTD 2013-04-03 CN claimed
CN-101588880-B Use of amine blends for foundry cores and foundry metals ARKEMA FRANCE 2012-03-07 CN claimed
CN-101323701-B Long glass fiber reinforced hard polyurethane synthetic material sleeper and method for preparing the same UNIV NANJING FORESTRY 2010-06-23 CN claimed
US-20100126690-A1 USE OF AMINE BLENDS FOR FOUNDRY SHAPED CORES AND CASTING METALS ARKEMA FRANCE (FR) 2010-05-27 US claimed
CN-101588880-A Use of amine blends for foundry cores and foundry metals ARKEMA FRANCE (FR) 2009-11-25 CN claimed
EP-2106310-A1 USE OF AMINE BLENDS FOR FOUNDRY SHAPED CORES AND CASTING METALS ARKEMA FRANCE (FR) 2009-10-07 EP claimed
CN-100530545-C Method for forming organic light-emitting layer MECHARONICS CO LTD (KR) 2009-08-19 CN claimed
CN-101323701-A Long glass fiber reinforced hard polyurethane synthetic material sleeper and method for preparing the same UNIV NANJING FORESTRY (CN) 2008-12-17 CN claimed
WO-2008090161-A1 USE OF AMINE BLENDS FOR FOUNDRY SHAPED CORES AND CASTING METALS ARKEMA FRANCE (FR) 2008-07-31 WO claimed