SCHEMBL28423930

SCHEMBL28423930

NC(=O)c1ccc(N[C@@H]2CCCNC2)c(N2CCOCC2)c1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 2/20 0.53
BTK Q06187 1/20 0.48
FLT3 P36888 10/20 0.47
CHEK1 O14757 5/20 0.44
KCNH2 Q12809 3/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28425526 0.81 KMT2A (0.52) IRAK4FLT3CHEK1KCNH2
SCHEMBL28419107 0.81 IRAK4 (0.50) IRAK4FLT3
SCHEMBL28420343 0.81 IRAK4 (0.49) IRAK4FLT3CHEK1KCNH2
SCHEMBL28418443 0.81 IRAK4 (0.49) IRAK4FLT3
SCHEMBL28424661 0.80 IRAK4 (0.52) IRAK4FLT3
SCHEMBL28416018 0.79 FLT3 (0.45) IRAK4FLT3ALDH1A1LMNA
SCHEMBL28423924 0.79 FLT3 (0.44) IRAK4FLT3
SCHEMBL28418539 0.79 IRAK4 (0.51) IRAK4FLT3KDM4EALDH1A1LMNA
SCHEMBL28422780 0.79 DDB1 (0.51) IRAK4FLT3KDM4E
SCHEMBL28418400 0.78 FLT3 (0.48) IRAK4FLT3ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111217816-B FLT3 kinase inhibitor and preparation and application thereof 中国科学院上海药物研究所 2022-08-16 CN disclosed
CN-111217816-A FLT3 kinase inhibitor and preparation and application thereof 中国科学院上海药物研究所 2020-06-02 CN disclosed