SCHEMBL28426727

SCHEMBL28426727

CC(=O)N[C@H]1CC[C@H](c2ccnc3ccccc32)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.46
MAPK8 P45983 2/20 0.46
MAPK9 P45984 2/20 0.46
MAPK10 P53779 2/20 0.46
CYP2C9 P11712 1/20 0.46
CCNE1 P24864 1/20 0.46
CDK2 P24941 1/20 0.46
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
PTK2B Q14289 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CAMKK1 Q8N5S9 1/20 0.42
CAMKK2 Q96RR4 1/20 0.42
DRD2 P14416 4/20 0.42
HTR2A P28223 4/20 0.42
DRD3 P35462 4/20 0.42
AR P10275 2/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21146433 0.82 IDO1 (0.43) IDO1CAMKK1CAMKK2DRD2HTR2A
SCHEMBL21052509 0.82 IDO1 (0.43) IDO1CAMKK1CAMKK2DRD2HTR2A
SCHEMBL21052508 0.82 IDO1 (0.43) IDO1CAMKK1CAMKK2DRD2HTR2A
SCHEMBL21146772 0.82 IDO1 (0.43) IDO1CAMKK1CAMKK2DRD2HTR2A
SCHEMBL29392938 0.81 MAPT (0.54) RAB9ANPC1TP53MAPTPTK2B
SCHEMBL17075123 0.81 MAPT (0.54) RAB9ANPC1TP53MAPTPTK2B
SCHEMBL22424952 0.81 P2RX7 (0.56) IDO1CYP2C9RAB9ATP53SMN1; SMN2
SCHEMBL22424964 0.81 P2RX7 (0.56) IDO1CYP2C9RAB9ATP53SMN1; SMN2
SCHEMBL21146333 0.81 P2RX7 (0.56) IDO1CYP2C9RAB9ATP53SMN1; SMN2
SCHEMBL28304231 0.79 NPY5R (0.45) IDO1CYP2C9RAB9ANPC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111417626-A Modulators of indoleamine2,3-dioxygenase 葛兰素史克知识产权开发有限公司 2020-07-14 CN disclosed