SCHEMBL28428367

SCHEMBL28428367

O=C(NS(=O)(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1nn(Cc2ccccc2)c2ccccc12

nearest known ligand 0.88

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 2/20 0.88
BCL2 P10415 3/20 0.53
VCAM1 P19320 3/20 0.53
BCL2L1 Q07817 1/20 0.51
PTGER4 P35408 5/20 0.48
SLC25A1 P53007 1/20 0.47
FBP1 P09467 1/20 0.46
DNMT1 P26358 1/20 0.45
DNMT3A Q9Y6K1 1/20 0.45
IDH1 O75874 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
PMP22 Q01453 1/20 0.43
HIF1A Q16665 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CCR2 P41597 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28431236 0.94 MCL1 (1.00) MCL1BCL2VCAM1BCL2L1PTGER4
SCHEMBL28423992 0.93 MCL1 (0.85) MCL1BCL2VCAM1BCL2L1PTGER4
SCHEMBL28421273 0.93 MCL1 (0.85) MCL1BCL2VCAM1BCL2L1PTGER4
SCHEMBL28429759 0.86 MCL1 (0.67) MCL1PTGER4IDH1
SCHEMBL28434112 0.84 MCL1 (0.84) MCL1BCL2PTGER4CCR2
SCHEMBL28424343 0.84 MCL1 (0.63) MCL1PTGER4CYP1A2CYP3A4CYP2D6
SCHEMBL28430356 0.79 MCL1 (0.65) MCL1PTGER4SMN1; SMN2
SCHEMBL28429765 0.79 MCL1 (0.65) MCL1PTGER4NPSR1SMN1; SMN2
SCHEMBL28424028 0.77 MCL1 (0.61) MCL1BCL2PTGER4
SCHEMBL28424695 0.77 MCL1 (0.61) MCL1BCL2PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111423379-A Substituted 3-indazole Mcl-1 protein inhibitor, preparation method and application 湖南科技大学 2020-07-17 CN claimed
CN-111423379-B Substituted 3-indazole Mcl-1 protein inhibitor, preparation method and application 湖南科技大学 2021-08-03 CN disclosed
CN-111423379-A Substituted 3-indazole Mcl-1 protein inhibitor, preparation method and application 湖南科技大学 2020-07-17 CN disclosed