SCHEMBL28429765

SCHEMBL28429765

Cc1ccc(Cn2nc(C(=O)NS(=O)(=O)c3ccc([N+](=O)[O-])cc3)c3ccccc32)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.65
PTGER4 P35408 4/20 0.46
P2RY14 Q15391 1/20 0.46
KMT2A Q03164 1/20 0.45
MMP1 P03956 1/20 0.45
MMP2 P08253 1/20 0.45
MMP9 P14780 1/20 0.45
MMP8 P22894 1/20 0.45
MMP13 P45452 1/20 0.45
CNR1 P21554 1/20 0.44
LMNA P02545 2/20 0.43
MITF O75030 1/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
FLT1 P17948 2/20 0.43
FLT4 P35916 2/20 0.43
KDR P35968 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28429759 0.92 MCL1 (0.67) MCL1PTGER4KMT2ACNR1FLT1
SCHEMBL28430356 0.91 MCL1 (0.65) MCL1PTGER4KMT2AMMP1MMP2
SCHEMBL28424028 0.88 MCL1 (0.61) MCL1PTGER4CNR1MAPTFLT1
SCHEMBL28434112 0.88 MCL1 (0.84) MCL1PTGER4FLT1FLT4KDR
SCHEMBL28421273 0.87 MCL1 (0.85) MCL1PTGER4CNR1LMNAMAPT
SCHEMBL24273075 0.83 MCL1 (0.61) MCL1PTGER4CNR1FLT1FLT4
SCHEMBL24273177 0.83 MCL1 (0.53) MCL1PTGER4KMT2ACNR1MAPT
SCHEMBL28424343 0.80 MCL1 (0.63) MCL1PTGER4KMT2ALMNAHTT
SCHEMBL28428367 0.79 MCL1 (0.88) MCL1PTGER4SMN1; SMN2NPSR1
SCHEMBL28431236 0.79 MCL1 (1.00) MCL1PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111423379-A Substituted 3-indazole Mcl-1 protein inhibitor, preparation method and application 湖南科技大学 2020-07-17 CN claimed
CN-111423379-B Substituted 3-indazole Mcl-1 protein inhibitor, preparation method and application 湖南科技大学 2021-08-03 CN disclosed
CN-111423379-A Substituted 3-indazole Mcl-1 protein inhibitor, preparation method and application 湖南科技大学 2020-07-17 CN disclosed