SCHEMBL28432151

SCHEMBL28432151

C=Cn1c(=O)[nH]c2nc[nH]c2c1=O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 9/20 0.61
ADORA3 P0DMS8 6/20 0.61
ADORA2A P29274 6/20 0.58
PDE4A P27815 4/20 0.54
PDE4B Q07343 4/20 0.54
PDE4C Q08493 4/20 0.54
PDE4D Q08499 4/20 0.54
ABL1 P00519 1/20 0.44
RIN1 Q13671 1/20 0.44
ACHE P22303 1/20 0.43
GDA Q9Y2T3 1/20 0.43
ADORA1 P30542 1/20 0.37
TDP1 Q9NUW8 2/20 0.36
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
PTGS1 P23219 1/20 0.35
HBB P68871 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28837899 0.85 ADORA2B (0.60) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL8536539 0.77 ADORA2B (0.55) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL6464355 0.76 ADORA2B (1.00) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL7491449 0.75 ADORA2B (0.56) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL5134361 0.75 ADORA2B (0.97) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL7170414 0.75 ADORA2B (0.52) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL7170406 0.75 ADORA2B (0.52) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL2842234 0.74 ADORA2B (0.55) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL7972790 0.74 ADORA2B (0.55) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL941656 0.74 ADORA2B (0.55) ADORA2BADORA3ADORA2APDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111333648-B 8-substituted aromatic ring vinyl xanthine derivative and application thereof 东莞市东阳光新药研发有限公司 2021-05-11 CN disclosed
CN-111333648-B 8-substituted aromatic ring vinyl xanthine derivative and application thereof 东莞市东阳光新药研发有限公司 2021-05-11 CN disclosed
CN-111333648-B 8-substituted aromatic ring vinyl xanthine derivative and application thereof 东莞市东阳光新药研发有限公司 2021-05-11 CN disclosed
CN-111333648-A 8-substituted aromatic ring vinyl xanthine derivative and application thereof 东莞市东阳光新药研发有限公司 2020-06-26 CN disclosed
CN-111333648-A 8-substituted aromatic ring vinyl xanthine derivative and application thereof 东莞市东阳光新药研发有限公司 2020-06-26 CN disclosed
CN-111333648-A 8-substituted aromatic ring vinyl xanthine derivative and application thereof 东莞市东阳光新药研发有限公司 2020-06-26 CN disclosed