SCHEMBL28434643

SCHEMBL28434643

FC(F)(F)C#Cc1ccc(-c2cccs2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.44
KCNH2 Q12809 2/20 0.43
CYP17A1 P05093 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
PDK2 Q15119 1/20 0.39
HRH3 Q9Y5N1 1/20 0.38
ERN1 O75460 2/20 0.37
LPL P06858 1/20 0.37
LIPG Q9Y5X9 1/20 0.37
PRMT6 Q96LA8 1/20 0.37
CYP2E1 P05181 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2A6 P11509 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2B6 P20813 1/20 0.37
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10300120 0.83 LTA4H (0.55) LTA4HKCNH2CYP17A1CYP11B1CYP11B2
SCHEMBL10300217 0.81 LTA4H (0.53) LTA4HKCNH2CYP17A1CYP11B1CYP11B2
SCHEMBL6852436 0.77 LTA4H (0.48) LTA4HKCNH2CYP17A1CYP11B1CYP11B2
SCHEMBL16473175 0.77 CYP1A1 (0.53) LTA4HKCNH2CYP17A1CYP11B1CYP11B2
SCHEMBL338810 0.74 LTA4H (0.70) LTA4HKCNH2CYP17A1CYP11B1CYP11B2
SCHEMBL28967308 0.74 APP (0.48) LTA4HKCNH2CYP17A1CYP11B1CYP11B2
SCHEMBL13247242 0.74 HDAC2 (0.54) LTA4HKCNH2CYP17A1CYP11B1CYP11B2
SCHEMBL154628 0.74 LTA4H (0.53) LTA4HKCNH2CYP17A1CYP11B1CYP11B2
SCHEMBL28440897 0.74 CYP1A2 (0.54) KCNH2CYP3A4MAPTALDH1A1TDP1
SCHEMBL6854037 0.72 LTA4H (0.44) LTA4HKCNH2CYP17A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111423304-B Synthetic method of 1,1-difluoroolefin compound 合肥工业大学 2023-02-28 CN disclosed
CN-111454286-A Synthetic method of difluoroalkenyl boron compound 合肥工业大学 2020-07-28 CN disclosed
CN-111423304-A Synthesis method of 1, 1-difluoroolefin compound 合肥工业大学 2020-07-17 CN disclosed