SCHEMBL28434877

SCHEMBL28434877

Cc1cccc2c1c(C)c(C(N)=O)n2C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 1/20 0.41
TSHR P16473 2/20 0.39
MAPT P10636 3/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
PKM P14618 1/20 0.38
IDO1 P14902 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
MDM2 Q00987 1/20 0.38
MCL1 Q07820 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
KDM4E B2RXH2 4/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PARP1 P09874 3/20 0.37
EGFR P00533 1/20 0.36
SRC P12931 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28263963 0.98 SLC9A1 (0.40) SLC9A1TSHRMAPTALDH1A1LMNA
Hydrochloric Acid SCHEMBL28262770 0.98 SLC9A1 (0.40) SLC9A1TSHRMAPTALDH1A1LMNA
SCHEMBL2662182 0.85 SLC9A1 (0.40) SLC9A1TSHRMAPTALDH1A1LMNA
SCHEMBL1253404 0.85 EGFR (0.42) SLC9A1TSHRMAPTALDH1A1LMNA
Hydrochloric Acid SCHEMBL1504224 0.84 EGFR (0.41) SLC9A1TSHRMAPTALDH1A1LMNA
SCHEMBL2662184 0.83 PARP1 (0.37) SLC9A1MAPTALDH1A1PKMMEN1
SCHEMBL28268477 0.77 EGFR (0.43) SLC9A1MAPTALDH1A1LMNAPKM
SCHEMBL6595214 0.76 TSHR (0.64) TSHRMAPTALDH1A1LMNAPKM
SCHEMBL35212204 0.76 TSHR (0.64) TSHRMAPTALDH1A1LMNAPKM
Hydrochloric Acid SCHEMBL28262758 0.75 TSHR (0.62) TSHRMAPTALDH1A1LMNAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111484484-B 2, 4-diaryl aminopyrimidine derivative containing aromatic heterocycle and preparation and application thereof 沈阳药科大学 2021-11-23 CN claimed
CN-111484484-A 2, 4-diaryl aminopyrimidine derivative containing aromatic heterocycle and preparation and application thereof 沈阳药科大学 2020-08-04 CN claimed
CN-111484484-B 2, 4-diaryl aminopyrimidine derivative containing aromatic heterocycle and preparation and application thereof 沈阳药科大学 2021-11-23 CN disclosed
CN-111484484-A 2, 4-diaryl aminopyrimidine derivative containing aromatic heterocycle and preparation and application thereof 沈阳药科大学 2020-08-04 CN disclosed