SCHEMBL2843906

SCHEMBL2843906

O=C(NO)C(c1ccccc1)N1CCOCC1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.65
CYP3A4 P08684 2/20 0.65
CYP2C19 P33261 2/20 0.65
TSHR P16473 4/20 0.64
LMNA P02545 3/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
GAA P10253 1/20 0.51
KCNA5 P22460 1/20 0.51
MMP8 P22894 1/20 0.50
ADRB2 P07550 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27777209 0.89 ALDH1A1 (0.67) ALDH1A1CYP3A4CYP2C19TSHRMMP8
SCHEMBL27798585 0.87 CYP3A4 (0.58) ALDH1A1CYP3A4CYP2C19TSHRLMNA
SCHEMBL1706030 0.85 ALDH1A1 (0.73) ALDH1A1CYP3A4CYP2C19TSHRLMNA
SCHEMBL627906 0.85 ALDH1A1 (0.73) ALDH1A1CYP3A4CYP2C19TSHRLMNA
SCHEMBL2846505 0.84 GAA (0.68) ALDH1A1CYP3A4CYP2C19TSHRLMNA
Hydrochloric Acid SCHEMBL15063255 0.83 ALDH1A1 (0.77) ALDH1A1CYP3A4CYP2C19TSHRLMNA
SCHEMBL2841585 0.83 NPY2R (0.51) ALDH1A1CYP3A4CYP2C19TSHRLMNA
SCHEMBL28839977 0.81 ALDH1A1 (0.58) ALDH1A1CYP3A4CYP2C19TSHRLMNA
SCHEMBL6598560 0.81 ALDH1A1 (0.68) ALDH1A1CYP3A4CYP2C19TSHRLMNA
SCHEMBL15711320 0.81 ALDH1A1 (0.68) ALDH1A1CYP3A4CYP2C19TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9096565-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2015-08-04 US disclosed
US-9096565-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2015-08-04 US disclosed
US-9096565-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2015-08-04 US disclosed
CN-101679220-A Histone deacetylase inhibitor METHYLGENE INC 2010-03-24 CN disclosed
EP-2139850-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2010-01-06 EP disclosed
US-20090181943-A1 Inhibitors of Histone Deacetylase METHYLGENE INC. (CA) 2009-07-16 US disclosed
US-20090181943-A1 Inhibitors of Histone Deacetylase METHYLGENE INC. (CA) 2009-07-16 US disclosed
US-20090181943-A1 Inhibitors of Histone Deacetylase METHYLGENE INC. (CA) 2009-07-16 US disclosed
WO-2008122115-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2008-10-16 WO disclosed
WO-2008122115-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2008-10-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090181943-A1 Inhibitors of Histone Deacetylase HDAC1, HDAC11, HDAC3 ALDH1A1 532/4885CYP3A4 1017/4885CYP2C19 782/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.