SCHEMBL28443180

SCHEMBL28443180

COC(=O)c1cccc2nnn(Cc3ccccc3)c12

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.56
CYP1A2 P05177 1/20 0.56
MAPK10 P53779 1/20 0.54
MAPK1 P28482 2/20 0.48
SLC9A1 P19634 1/20 0.48
GRM2 Q14416 1/20 0.48
CYP19A1 P11511 4/20 0.47
HPGD P15428 4/20 0.46
ALDH1A1 P00352 3/20 0.46
TSHR P16473 2/20 0.46
KMT2A Q03164 2/20 0.45
KDM4E B2RXH2 1/20 0.45
USP2 O75604 1/20 0.45
HSD17B10 Q99714 1/20 0.45
HCAR3 P49019 2/20 0.45
LMNA P02545 1/20 0.43
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1271587 0.91 TDP1 (0.50) SMN1; SMN2CYP1A2MAPK10MAPK1CYP19A1
SCHEMBL28897969 0.88 NPC1 (0.50) SMN1; SMN2CYP1A2MAPK10MAPK1HPGD
SCHEMBL28450969 0.85 GRM2 (0.54) SLC9A1GRM2CYP19A1HPGDALDH1A1
SCHEMBL28443265 0.80 CYP1A2 (0.54) SMN1; SMN2CYP1A2MAPK10MAPK1CYP19A1
SCHEMBL12900276 0.77 TDP1 (0.55) SLC9A1GRM2CYP19A1HPGDHCAR3
SCHEMBL28451005 0.77 RECQL (0.48) SMN1; SMN2CYP1A2ALDH1A1TSHRKMT2A
SCHEMBL28440773 0.77 CYP11B1 (0.48) SMN1; SMN2MAPK10TSHRKMT2AKDM4E
SCHEMBL2014506 0.76 KDM4E (0.43) SMN1; SMN2CYP1A2SLC9A1ALDH1A1TSHR
SCHEMBL11769430 0.75 CYP1A2 (0.51) SMN1; SMN2CYP1A2MAPK10MAPK1CYP19A1
SCHEMBL11767746 0.75 SMN1; SMN2 (0.57) SMN1; SMN2CYP1A2MAPK1CYP19A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111606928-A Azacyclodiketone compound and preparation method thereof 维清生物科技(上海)有限公司 2020-09-01 CN disclosed