SCHEMBL28443265

SCHEMBL28443265

COC(=O)c1ccc(F)c2nnn(Cc3ccccc3)c12

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
FGFR1 P11362 1/20 0.48
FGFR4 P22455 1/20 0.48
ADORA3 P0DMS8 2/20 0.44
HPGD P15428 3/20 0.44
TP53 P04637 2/20 0.44
ALDH1A1 P00352 2/20 0.44
TSHR P16473 2/20 0.44
CYP19A1 P11511 2/20 0.43
KMT2A Q03164 3/20 0.42
KDM4E B2RXH2 1/20 0.42
USP2 O75604 1/20 0.42
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MEN1 O00255 1/20 0.42
ATM Q13315 1/20 0.42
MAPK10 P53779 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28454653 0.86 HPGD (0.49) CYP1A2SMN1; SMN2ADORA3HPGDTP53
SCHEMBL11769430 0.80 CYP1A2 (0.51) CYP1A2SMN1; SMN2FGFR1FGFR4ADORA3
SCHEMBL11767746 0.80 SMN1; SMN2 (0.57) CYP1A2SMN1; SMN2ADORA3HPGDTP53
SCHEMBL28443180 0.80 SMN1; SMN2 (0.56) CYP1A2SMN1; SMN2HPGDALDH1A1TSHR
SCHEMBL28450982 0.80 SMN1; SMN2 (0.44) CYP1A2SMN1; SMN2TP53ALDH1A1TSHR
SCHEMBL11772597 0.78 CYP1A2 (0.52) CYP1A2SMN1; SMN2ADORA3HPGDALDH1A1
SCHEMBL11770744 0.78 CYP1A2 (0.48) CYP1A2SMN1; SMN2ADORA3HPGDALDH1A1
SCHEMBL11770739 0.77 CYP1A2 (0.50) CYP1A2SMN1; SMN2FGFR1FGFR4HPGD
SCHEMBL28447631 0.73 GRM2 (0.56) ADORA3TP53ALDH1A1TSHRKMT2A
SCHEMBL11769893 0.73 CYP1A2 (0.43) CYP1A2SMN1; SMN2ADORA3HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111606928-A Azacyclodiketone compound and preparation method thereof 维清生物科技(上海)有限公司 2020-09-01 CN disclosed