SCHEMBL2844447

SCHEMBL2844447

CC1CCN(C(Cc2ccc(C(C)C(=O)O)cc2-c2ccc(C(F)(F)F)cc2)c2ccc(F)c(F)c2)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.61
PTGS2 P35354 3/20 0.61
KCNH2 Q12809 2/20 0.61
PSEN1 P49768 2/20 0.61
PSEN2 P49810 2/20 0.61
APH1B Q8WW43 2/20 0.61
NCSTN Q92542 2/20 0.61
APH1A Q96BI3 2/20 0.61
PSENEN Q9NZ42 2/20 0.61
AKR1C3 P42330 8/20 0.53
AKR1C2 P52895 8/20 0.53
TRPV1 Q8NER1 4/20 0.42
APP P05067 3/20 0.41
TACR1 P25103 1/20 0.40
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP3A4 P08684 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
FABP2 P12104 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2847511 0.76 KCNH2 (1.00) PTGS1PTGS2KCNH2PSEN1PSEN2
SCHEMBL24913685 0.76 KCNH2 (1.00) PTGS1PTGS2KCNH2PSEN1PSEN2
SCHEMBL2846664 0.76 KCNH2 (1.00) PTGS1PTGS2KCNH2PSEN1PSEN2
SCHEMBL2848167 0.72 AKR1C3 (0.66) PTGS1PTGS2KCNH2PSEN1PSEN2
SCHEMBL2846830 0.72 KCNH2 (0.68) PTGS1PTGS2KCNH2PSEN1PSEN2
SCHEMBL1372793 0.72 AKR1C3 (1.00) PTGS1PTGS2PSEN1PSEN2APH1B
SCHEMBL2848843 0.71 KCNH2 (0.59) PTGS1PTGS2KCNH2PSEN1PSEN2
SCHEMBL2844333 0.70 AKR1C3 (0.59) PTGS1PTGS2KCNH2PSEN1PSEN2
SCHEMBL2844065 0.67 KCNH2 (0.82) PTGS1PTGS2KCNH2PSEN1PSEN2
SCHEMBL2878421 0.67 KCNH2 (0.77) PTGS1PTGS2KCNH2PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010138901-A1 CARBOXYLIC ACID-CONTAINING COMPOUNDS, DERIVATIVES THEREOF, AND RELATED METHODS OF USE BIOGEN IDEC MA INC (US) 2010-12-02 WO claimed