SCHEMBL28447693

SCHEMBL28447693

COc1cc(Cl)c(N)cc1Nc1ncc(Cl)c(Nc2ccc(N3CCOCC3)cc2OC)n1

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 13/20 0.85
INSR P06213 8/20 0.85
LRRK2 Q5S007 3/20 0.76
MAPK8 P45983 2/20 0.73
MAPK9 P45984 2/20 0.73
MAPK10 P53779 2/20 0.73
EGFR P00533 2/20 0.70
IGF1R P08069 2/20 0.70
CDC7 O00311 1/20 0.70
PLK4 O00444 1/20 0.70
CHEK1 O14757 1/20 0.70
AURKA O14965 1/20 0.70
DCLK1 O15075 1/20 0.70
PDPK1 O15530 1/20 0.70
DAPK3 O43293 1/20 0.70
DYRK3 O43781 1/20 0.70
JAK2 O60674 1/20 0.70
PRKD3 O94806 1/20 0.70
PAK4 O96013 1/20 0.70
CHEK2 O96017 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28054061 0.92 ALK (0.81) ALKINSRLRRK2MAPK8MAPK9
SCHEMBL29435444 0.90 ALK (0.84) ALKINSRLRRK2MAPK8MAPK9
SCHEMBL22087543 0.90 ALK (0.84) ALKINSRLRRK2MAPK8MAPK9
SCHEMBL12311873 0.87 LRRK2 (1.00) ALKINSRLRRK2MAPK8MAPK9
SCHEMBL18650996 0.85 ALK (0.85) ALKINSRLRRK2MAPK8MAPK9
SCHEMBL11916449 0.85 ALK (0.84) ALKINSRLRRK2MAPK8MAPK9
SCHEMBL2061740 0.84 ALK (0.91) ALKINSRLRRK2MAPK8MAPK9
SCHEMBL375436 0.84 MAPK9 (0.86) ALKINSRLRRK2MAPK8MAPK9
SCHEMBL2060832 0.83 ALK (0.82) ALKINSRLRRK2MAPK8MAPK9
SCHEMBL31174591 0.83 ALK (0.87) ALKINSRLRRK2MAPK8MAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384694-B Substituted aminopyrimidine derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2020-09-04 CN disclosed