SCHEMBL28447992

SCHEMBL28447992

O=[N+]([O-])c1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2cc1OCCN1CCOCC1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.74
ERBB2 P04626 4/20 0.69
KDR P35968 3/20 0.69
EPHB4 P54760 3/20 0.69
KIT P10721 3/20 0.69
SRC P12931 3/20 0.69
ERBB3 P21860 3/20 0.69
ERBB4 Q15303 3/20 0.69
CIT O14578 2/20 0.69
GAK O14976 2/20 0.69
EPHB6 O15197 2/20 0.69
RIPK2 O43353 2/20 0.69
STK17B O94768 2/20 0.69
STK10 O94804 2/20 0.69
ABL1 P00519 2/20 0.69
LCK P06239 2/20 0.69
LYN P07948 2/20 0.69
RET P07949 2/20 0.69
MET P08581 2/20 0.69
HCK P08631 2/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5675006 0.96 EGFR (0.75) EGFRERBB2KDREPHB4KIT
SCHEMBL7003295 0.91 EGFR (0.68) EGFRERBB2KDREPHB4KIT
SCHEMBL28935220 0.89 EGFR (0.92) EGFRERBB2KDREPHB4KIT
SCHEMBL29577309 0.89 EGFR (0.92) EGFRERBB2KDREPHB4KIT
SCHEMBL31193424 0.89 EGFR (0.65) EGFRERBB2KDREPHB4KIT
SCHEMBL3590411 0.89 EGFR (0.71) EGFRERBB2KDREPHB4KIT
SCHEMBL31193415 0.87 EGFR (0.77) EGFRERBB2
SCHEMBL7002698 0.87 EGFR (0.74) EGFRERBB2KDREPHB4KIT
SCHEMBL7003865 0.86 EGFR (0.70) EGFRERBB2KDREPHB4KIT
SCHEMBL29087952 0.85 KDR (0.56) EGFRKDREPHB4SRCLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107556295-B Quinazoline derivatives and process for their preparation 正大天晴药业集团股份有限公司 2020-09-04 CN disclosed