SCHEMBL28448563

SCHEMBL28448563

COc1cc(N(C)CCN(C)C)c([N+](=O)[O-])cc1Nc1nc(N)c(Cl)c(-c2ccc(N3CCOCC3)cc2OC)n1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.47
ALK Q9UM73 7/20 0.41
INSR P06213 4/20 0.41
KCNH2 Q12809 3/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
LRRK2 Q5S007 1/20 0.40
IGF1R P08069 2/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
FGFR3 P22607 1/20 0.38
MAPK8 P45983 1/20 0.38
MAPK9 P45984 1/20 0.38
MAPK10 P53779 1/20 0.38
TTK P33981 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28455448 0.86 ALK (0.46) EGFRALKINSRKCNH2LRRK2
SCHEMBL28448564 0.82 EGFR (0.44) EGFRKCNH2IGF1R
SCHEMBL28053863 0.81 ALK (0.66) EGFRALKINSRKCNH2CYP3A4
SCHEMBL17059196 0.77 EGFR (0.52) EGFRALKINSRKCNH2CYP3A4
SCHEMBL17059199 0.76 EGFR (0.52) EGFRALKINSRKCNH2CYP3A4
SCHEMBL29855954 0.71 EGFR (0.54) EGFRALK
SCHEMBL28053984 0.70 ALK (0.58) EGFRALKINSRKCNH2CYP3A4
SCHEMBL18239603 0.69 EGFR (0.74) EGFRINSRKCNH2IGF1R
SCHEMBL30041502 0.69 EGFR (0.51) EGFRALKKCNH2
SCHEMBL14719261 0.68 EGFR (0.74) EGFRINSRKCNH2IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384694-B Substituted aminopyrimidine derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2020-09-04 CN disclosed