SCHEMBL28449100

SCHEMBL28449100

O=C(O)C1CN(c2ncccn2)C1

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.68
CYP2C19 P33261 1/20 0.68
TSHR P16473 2/20 0.46
ALDH1A1 P00352 1/20 0.46
NOTUM Q6P988 3/20 0.44
SLC6A7 Q99884 1/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 2/20 0.42
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HPGD P15428 1/20 0.42
GAA P10253 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
MDM2 Q00987 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15416556 0.85 KDM4E (0.81) KDM4ECYP2C19TSHRALDH1A1NOTUM
SCHEMBL195842 0.81 KDM4E (1.00) KDM4ECYP2C19ALDH1A1NOTUMLMNA
SCHEMBL16302107 0.79 KDM4E (0.45) KDM4ECYP2C19ALDH1A1NOTUMHSD17B10
SCHEMBL17234262 0.78 GRIN2B (0.54) KDM4ECYP2C19TSHRALDH1A1NOTUM
SCHEMBL3585722 0.78 KDM4E (0.50) KDM4ECYP2C19TSHRALDH1A1LMNA
SCHEMBL21061696 0.78 KDM4E (0.47) KDM4ECYP2C19TSHRALDH1A1LMNA
SCHEMBL21151895 0.77 KDM4E (0.42) KDM4ECYP2C19ALDH1A1NOTUMHSD17B10
SCHEMBL29364193 0.76 SLC6A7 (0.50) KDM4ECYP2C19SLC6A7
SCHEMBL3575820 0.76 SLC6A7 (0.58) KDM4ETSHRALDH1A1SLC6A7MAPK1
SCHEMBL16433993 0.75 NOTUM (0.49) KDM4ECYP2C19NOTUMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116322692-A Autotaxin inhibitor compounds 日东制药株式会社 2023-06-23 CN disclosed
CN-111479813-B Triazolobenzazepines as vasopressin V1A receptor antagonists 吉瑞工厂 2023-03-21 CN disclosed
CN-111479813-A Triazolobenzazepines as vasopressin V1A receptor antagonists 吉瑞工厂 2020-07-31 CN disclosed